Inhibition of LZIP-mediated transcription through direct interaction with a novel host cell factor-like protein

J Biol Chem. 2001 Aug 3;276(31):28933-8. doi: 10.1074/jbc.M103893200. Epub 2001 May 30.

Abstract

Host cell factor 1 (HCF-1) is a cellular transcriptional coactivator which coordinates the assembly of enhancer complex through direct interactions with viral and cellular trans-activators such as VP16, Oct-1, LZIP, and GA-binding protein. These interactions are mediated by the beta-propeller domain comprising the first 380 residues of HCF-1 with six kelch repeats. Here we describe the identification and characterization of a novel HCF-like kelch repeat protein, designated HCLP-1. HCLP-1 is a ubiquitously expressed nuclear protein which is composed almost entirely of a six-bladed beta-propeller. HCLP-1 selectively interacts with LZIP but not with VP16. The physical interaction between HCLP-1 and LZIP leads to the repression of the LZIP-dependent transcription. The HCLP-1-binding domain of LZIP maps to residues 109-315, which contain the bZIP DNA-binding motif. Electrophoretic mobility shift assay demonstrates that HCLP-1 indeed interferes with the binding of LZIP to its DNA target. Thus, HCLP-1 serves a transcriptional co-repressor function mediated through its inhibitory interaction with the LZIP transcription factor. Our findings suggest a new mechanism for transcriptional regulation by HCF-like proteins.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Antigens, Neoplasm
  • Binding Sites
  • Conserved Sequence
  • Cyclic AMP Response Element-Binding Protein
  • DNA / chemistry
  • DNA / metabolism
  • DNA-Binding Proteins / metabolism
  • Gene Expression Regulation*
  • Genes, Reporter
  • HeLa Cells
  • Host Cell Factor C1
  • Humans
  • Kinetics
  • Leucine Zippers
  • Luciferases / genetics
  • Molecular Sequence Data
  • Protein Structure, Secondary
  • Proteins / chemistry*
  • Proteins / metabolism*
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism
  • Repetitive Sequences, Amino Acid
  • Sequence Alignment
  • Sequence Homology, Amino Acid
  • Transcription Factors / chemistry*
  • Transcription Factors / metabolism*
  • Transcription, Genetic*
  • Transfection

Substances

  • Antigens, Neoplasm
  • CREB3 protein, human
  • Cyclic AMP Response Element-Binding Protein
  • DNA-Binding Proteins
  • HCFC1 protein, human
  • Host Cell Factor C1
  • KLHDC2 protein, human
  • Proteins
  • Recombinant Proteins
  • Transcription Factors
  • DNA
  • Luciferases

Associated data

  • GENBANK/AF113131