Separate SCF(CDC4) recognition elements target Cdc6 for proteolysis in S phase and mitosis

EMBO J. 2001 Sep 3;20(17):4836-45. doi: 10.1093/emboj/20.17.4836.

Abstract

The Cdc6 DNA replication initiation factor is targeted for ubiquitin-mediated proteolysis by the E3 ubiquitin ligase SCF(CDC4) from the end of G1phase until mitosis in the budding yeast Saccharomyces cerevisiae. Here we describe a dominant-negative CDC6 mutant that, when overexpressed, arrests the cell cycle by inhibiting cyclin-dependent kinases (CDKs) and, thus, prevents passage through mitosis. This mutant protein inhibits CDKs more efficiently than wild-type Cdc6, in part because it is completely refractory to SCF(CDC4)-mediated proteolysis late in the cell cycle and consequently accumulates to high levels. The mutation responsible for this phenotype destroys a putative CDK phosphorylation site near the middle of the Cdc6 primary amino acid sequence. We show that this site lies within a novel Cdc4-interacting domain distinct from a Cdc4-interacting site identified previously near the N-terminus of the protein. We show that both sites can target Cdc6 for proteolysis in late G1/early S phase whilst only the newly identified site can target Cdc6 for proteolysis during mitosis.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Base Sequence
  • Binding Sites
  • Cell Cycle / drug effects
  • Cell Cycle / physiology*
  • Cell Cycle Proteins / chemistry
  • Cell Cycle Proteins / genetics
  • Cell Cycle Proteins / metabolism*
  • Cyclin-Dependent Kinases / metabolism
  • DNA Primers
  • F-Box Proteins*
  • Fungal Proteins / genetics
  • Fungal Proteins / metabolism
  • Galactose / metabolism
  • Genotype
  • Glucose / metabolism
  • Mitosis / physiology
  • Nocodazole / pharmacology
  • Phosphorylation
  • Promoter Regions, Genetic
  • S Phase / physiology
  • Saccharomyces cerevisiae / cytology*
  • Saccharomyces cerevisiae / genetics
  • Saccharomyces cerevisiae / growth & development
  • Saccharomyces cerevisiae Proteins*
  • Sequence Alignment
  • Sequence Homology, Amino Acid
  • Suppression, Genetic
  • Ubiquitin-Protein Ligases*

Substances

  • CDC4 protein, S cerevisiae
  • CDC6 protein, S cerevisiae
  • Cell Cycle Proteins
  • DNA Primers
  • F-Box Proteins
  • Fungal Proteins
  • Saccharomyces cerevisiae Proteins
  • Ubiquitin-Protein Ligases
  • Cyclin-Dependent Kinases
  • Glucose
  • Nocodazole
  • Galactose