Structure-activity relationship studies of isoquinolinone type anticancer agent

Arch Pharm Res. 2001 Aug;24(4):276-80. doi: 10.1007/BF02975091.

Abstract

Substituted isoquinolin-1-ones (1) were synthesized to test their in vitro anticancer activity. 3-Biphenyl-N-methylisoquinolin-1-one (7) showed the most potent anticancer activity against five different human cancer cell lines.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / chemical synthesis*
  • Antineoplastic Agents / pharmacology*
  • Drug Screening Assays, Antitumor
  • Humans
  • Indicators and Reagents
  • Isoquinolines / chemical synthesis*
  • Isoquinolines / pharmacology*
  • Magnetic Resonance Spectroscopy
  • Structure-Activity Relationship
  • Tumor Cells, Cultured

Substances

  • Antineoplastic Agents
  • Indicators and Reagents
  • Isoquinolines