Inhibition of mannose-binding lectin reduces postischemic myocardial reperfusion injury

Circulation. 2001 Sep 18;104(12):1413-8. doi: 10.1161/hc3601.095578.

Abstract

Background: Complement consists of a complex cascade of proteins involved in innate and adaptive immunity. The cascade can be activated through 3 distinct mechanisms, designated the classical, alternative, and lectin pathways. Although complement is widely accepted as participating in the pathophysiology of ischemia-reperfusion injury, the specific role of the lectin pathway has not been addressed.

Methods and results: Monoclonal antibodies (mAbs; P7E4 and 14C3.74, IgG1kappa isotypes) were raised against rat mannose-binding lectin (rMBL). Both mAbs recognized rMBL-A by Western analysis or surface plasmon resonance. P7E4, but not 14C3.74, exhibited a concentration-dependent inhibition of the lectin pathway, with maximal effect at 10 microg/mL. In vivo, rats were subjected to 30 minutes of left coronary artery occlusion and 4 hours of reperfusion. Complement C3 deposition was greatly attenuated in hearts pretreated with P7E4 compared with 14C3.74-treated hearts. Pretreatment with P7E4 (1 mg/kg) significantly reduced myocardial creatine kinase loss (48%), infarct size (39%), and neutrophil infiltration (47%) compared with 14C3.74-treated animals. In addition, P7E4 pretreatment significantly attenuated the expression of proinflammatory genes (intercellular adhesion molecule-1, vascular cell adhesion molecule-1, and interleukin-6) after ischemia-reperfusion.

Conclusions: The lectin complement pathway is activated after myocardial ischemia-reperfusion and leads to tissue injury. Blockade of the lectin pathway with inhibitory mAbs protects the heart from ischemia-reperfusion by reducing neutrophil infiltration and attenuating proinflammatory gene expression.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibodies, Monoclonal / metabolism
  • Antibodies, Monoclonal / pharmacology
  • Antibody Specificity
  • Carrier Proteins / antagonists & inhibitors*
  • Carrier Proteins / pharmacology
  • Cell Adhesion Molecules / biosynthesis
  • Cell Adhesion Molecules / genetics
  • Collectins
  • Complement Activation / drug effects
  • Complement C3 / metabolism
  • Creatine Kinase / metabolism
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Interleukins / biosynthesis
  • Interleukins / genetics
  • Male
  • Mannose / pharmacology
  • Monokines / biosynthesis
  • Monokines / genetics
  • Myocardial Ischemia / complications
  • Myocardial Ischemia / metabolism
  • Myocardial Ischemia / pathology
  • Myocardial Reperfusion Injury / etiology
  • Myocardial Reperfusion Injury / pathology
  • Myocardial Reperfusion Injury / prevention & control*
  • Myocardium / metabolism
  • Myocardium / pathology
  • Peroxidase / metabolism
  • RNA, Messenger / biosynthesis
  • Rats
  • Rats, Sprague-Dawley
  • Signal Transduction / drug effects
  • Surface Plasmon Resonance

Substances

  • Antibodies, Monoclonal
  • Carrier Proteins
  • Cell Adhesion Molecules
  • Collectins
  • Complement C3
  • Interleukins
  • Monokines
  • RNA, Messenger
  • Peroxidase
  • Creatine Kinase
  • Mannose