Self-association of model transmembrane alpha-helices is modulated by lipid structure

Biochemistry. 2001 Oct 16;40(41):12379-86. doi: 10.1021/bi011075y.

Abstract

We have developed a fluorescence quenching method using peptides containing 3,5-dibromotryrosine to measure oligomerization of model transmembrane alpha-helices in lipid bilayers. Peptides of the type Ac-LysLysGlyLeu(m)XLeu(n)LysLysAla-amide where X is tryptophan or 3,5-dibromotyrosine were found to form heterodimers in bilayers of phosphatidylcholine in the liquid-crystalline phase. The free energy of dimer formation changed little with increasing number of Leu residues from 16 to 22 but increased with increasing phospholipid fatty acyl chain length, with a slope of about 0.5 kJ mol(-1) per fatty acyl chain carbon. Peptides were excluded from lipid in the gel phase, resulting in increased levels of oligomerization. Addition of cholesterol to form the liquid-ordered state led to increased dimerization but without phase separation. The presence of phosphatidylethanolamine had little effect on dimerization.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Dimerization
  • Fluorescence
  • Gels
  • In Vitro Techniques
  • Lipid Bilayers / chemistry*
  • Membrane Proteins / chemistry*
  • Membranes, Artificial
  • Models, Molecular
  • Peptides / chemistry
  • Protein Structure, Secondary
  • Thermodynamics
  • Tyrosine / analogs & derivatives
  • Tyrosine / chemistry

Substances

  • Gels
  • Lipid Bilayers
  • Membrane Proteins
  • Membranes, Artificial
  • Peptides
  • Tyrosine
  • 3,5-dibromotyrosine