Signaling to the nucleus by an L-type calcium channel-calmodulin complex through the MAP kinase pathway

Science. 2001 Oct 12;294(5541):333-9. doi: 10.1126/science.1063395.

Abstract

Increases in the intracellular concentration of calcium ([Ca2+]i) activate various signaling pathways that lead to the expression of genes that are essential for dendritic development, neuronal survival, and synaptic plasticity. The mode of Ca2+ entry into a neuron plays a key role in determining which signaling pathways are activated and thus specifies the cellular response to Ca2+. Ca2+ influx through L-type voltage-activated channels (LTCs) is particularly effective at activating transcription factors such as CREB and MEF-2. We developed a functional knock-in technique to investigate the features of LTCs that specifically couple them to the signaling pathways that regulate gene expression. We found that an isoleucine-glutamine ("IQ") motif in the carboxyl terminus of the LTC that binds Ca2+-calmodulin (CaM) is critical for conveying the Ca2+ signal to the nucleus. Ca2+-CaM binding to the LTC was necessary for activation of the Ras/mitogen-activated protein kinase (MAPK) pathway, which conveys local Ca2+ signals from the mouth of the LTC to the nucleus. CaM functions as a local Ca2+ sensor at the mouth of the LTC that activates the MAPK pathway and leads to the stimulation of genes that are essential for neuronal survival and plasticity.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Motifs
  • Amino Acid Sequence
  • Animals
  • Calcium / metabolism*
  • Calcium Channels, L-Type / chemistry
  • Calcium Channels, L-Type / genetics
  • Calcium Channels, L-Type / metabolism*
  • Calcium Signaling
  • Calmodulin / metabolism*
  • Cell Membrane / metabolism
  • Cell Nucleus / metabolism*
  • Cells, Cultured
  • Cerebral Cortex / cytology
  • Cyclic AMP Response Element-Binding Protein / metabolism
  • DNA-Binding Proteins / metabolism
  • Enzyme Activation
  • Gene Expression Regulation
  • MAP Kinase Signaling System*
  • MEF2 Transcription Factors
  • Mitogen-Activated Protein Kinases / metabolism
  • Molecular Sequence Data
  • Mutation
  • Myogenic Regulatory Factors
  • Neurons / metabolism*
  • Phosphorylation
  • Phosphoserine / metabolism
  • Protein Structure, Tertiary
  • Rats
  • Rats, Long-Evans
  • Transcription Factors / metabolism
  • Transcription, Genetic
  • Transfection

Substances

  • Calcium Channels, L-Type
  • Calmodulin
  • Cyclic AMP Response Element-Binding Protein
  • DNA-Binding Proteins
  • MEF2 Transcription Factors
  • Myogenic Regulatory Factors
  • Transcription Factors
  • Phosphoserine
  • Mitogen-Activated Protein Kinases
  • Calcium