8-Prenylnaringenin, the phytoestrogen in hops and beer, upregulates the function of the E-cadherin/catenin complex in human mammary carcinoma cells

Eur J Cell Biol. 2001 Sep;80(9):580-5. doi: 10.1078/0171-9335-00190.

Abstract

The E-cadherin/catenin complex is a powerful invasion suppressor in epithelial cells. It is expressed in the human MCF-7 breast cancer cell line family, but functionally defective in the invasive MCF-7/6 variant. Previous experiments have shown that IGF-I, tamoxifen, retinoic acid and tangeretin are able to upregulate the function of this complex in MCF-7/6 cells. We investigated the effect of 8-prenylnaringenin (8-PN), the phytoestrogen present in hops and beer, on aggregation, growth and invasion in MCF-7/6 cells. 8-PN was found to stimulate E-cadherin-dependent aggregation and growth of MCF-7/6 cells in suspension. These effects could be inhibited by the pure anti-estrogen ICI 182,780. 8-PN did not affect invasion of MCF-7/6 cells in the chick heart assay in vitro. In all these aspects 8-PN mimics the effects of 17beta-estradiol on MCF-7/6 cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Beer*
  • Breast Neoplasms
  • Cadherins / metabolism*
  • Cell Adhesion / drug effects*
  • Cell Aggregation / drug effects*
  • Estrogens, Non-Steroidal / pharmacology*
  • Female
  • Flavanones*
  • Flavonoids / pharmacology*
  • Humans
  • Humulus / chemistry*
  • Isoflavones*
  • Phytoestrogens
  • Plant Preparations
  • Tumor Cells, Cultured
  • Tumor Stem Cell Assay
  • Up-Regulation

Substances

  • 8-prenylnaringenin
  • Cadherins
  • Estrogens, Non-Steroidal
  • Flavanones
  • Flavonoids
  • Isoflavones
  • Phytoestrogens
  • Plant Preparations