Administration of two antagonists of the cholecystokinin(B)/gastrin receptor does not totally inhibit the pancreatic response to a meal in the pig

Pancreas. 2002 Jan;24(1):47-52. doi: 10.1097/00006676-200201000-00007.

Abstract

Introduction and aims: The role of the cholecystokinin B (CCK(B))/gastrin receptor in the pancreatic response to a standard meal was investigated in the pig.

Methodology: Twenty-four pigs were prepared surgically for the collection of the pancreatic juice and an intravenous perfusion. On experimental days, the pigs were perfused with one of two CCK(B)antagonists (L-365,260 or PD 135156) or the vehicle for 2 hours. We offered them a standard meal 30 minutes after the beginning of the perfusion. The pancreatic secretion was collected for 4 hours starting 30 minutes before the perfusion. Its volume was recorded, and the protein concentrations were assayed.

Results: Neither antagonist totally abolished the postprandial peak of the pancreatic protein.

Conclusions: We suggest that the stimulation of pancreatic protein secretion by a meal is not mediated by CCK(B)/gastrin receptors. Because we previously showed that the CCK(A)receptor antagonist MK329 was no more able to abolish this response, CCK is probably not responsible for this response.

MeSH terms

  • Animals
  • Benzodiazepinones / pharmacology*
  • Dipeptides / pharmacology*
  • Dose-Response Relationship, Drug
  • Eating*
  • Male
  • Models, Animal
  • Pancreas / drug effects*
  • Pancreas / metabolism
  • Perfusion
  • Phenylurea Compounds / pharmacology*
  • Postprandial Period
  • Receptors, Cholecystokinin / antagonists & inhibitors*
  • Swine

Substances

  • Benzodiazepinones
  • Dipeptides
  • PD 135156
  • Phenylurea Compounds
  • Receptors, Cholecystokinin
  • L 365260