Gramicidin derivatives as membrane-based pH sensors

Biochim Biophys Acta. 2002 Jan 2;1558(1):26-33. doi: 10.1016/s0005-2736(01)00415-1.

Abstract

Ion channels provide a means for sensitive pH measurement at membrane interfaces. Detailed knowledge of the structure and function of gramicidin channels permits the engineering of pH-sensitive derivatives. Two derivatives, gramicidin-ethylenediamine and gramicidin-histamine, are shown to exhibit pH-dependent single-channel behaviour over the pH ranges 9-11 and 6.5-8.5, respectively. Thermal isomerization of a carbamate group at the entrance of the channels leads to a pattern of steps in single-channel recordings. The size of the steps depends on the time-averaged degree of protonation of the appended group (ethylenediamine or histamine). Measurement of the size of the steps thus permits single-molecule pH sensing under symmetrical pH conditions or in the presence of a pH gradient.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biosensing Techniques*
  • Cell Membrane / chemistry*
  • Ethylenediamines / chemistry
  • Gramicidin / chemistry*
  • Histamine / chemistry
  • Hydrogen-Ion Concentration
  • Ion Channels / chemistry
  • Molecular Structure

Substances

  • Ethylenediamines
  • Ion Channels
  • Gramicidin
  • ethylenediamine
  • Histamine