Chromium treatment decreases the sensitivity of 5-HT2A receptors

Psychopharmacology (Berl). 2002 Feb;159(4):432-6. doi: 10.1007/s00213-001-0960-7. Epub 2001 Nov 28.

Abstract

Rationale: Recent case series suggest that chromium picolinate in doses of 400 microg daily may have antidepressant properties, perhaps through increasing the peripheral availability of tryptophan for brain serotonin (5-HT) synthesis.

Objectives: To determine the effects of chromium treatment on plasma tryptophan availability and on brain 5-HT function in human and animal models.

Methods: We studied the effects of short-term chromium supplementation on plasma concentrations of tryptophan and other large neutral amino acids. Brain 5-HT function was assessed by measuring the corticosterone/cortisol response to the 5-HT precursor, 5-hydroxytryptophan (5-HTP), a response believed to be mediated via indirect activation of 5-HT(2A) receptors.

Results: In rats, chromium increased peripheral and central tryptophan availability and elevated brain 5-HT content. Changes in peripheral tryptophan availability were not seen in humans but in both rats and humans, chromium lowered the cortisol response to challenge with 5-HTP.

Conclusions: Chromium can modify brain 5-HT function in humans and animals, perhaps by altering the sensitivity of central 5-HT(2A) receptors.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Analysis of Variance
  • Animals
  • Brain / drug effects
  • Brain / metabolism
  • Chromium / pharmacology*
  • Corticosterone / blood
  • Cross-Over Studies
  • Female
  • Humans
  • Male
  • Middle Aged
  • Rats
  • Rats, Sprague-Dawley
  • Receptor, Serotonin, 5-HT2A
  • Receptors, Serotonin / metabolism*
  • Serotonin / metabolism
  • Single-Blind Method
  • Tryptophan / blood

Substances

  • Receptor, Serotonin, 5-HT2A
  • Receptors, Serotonin
  • Chromium
  • Serotonin
  • Tryptophan
  • Corticosterone