A minimal receptor-Ig chimera of human FcepsilonRI alpha-chain efficiently binds secretory and membrane IgE

Protein Eng. 2002 Jan;15(1):51-7. doi: 10.1093/protein/15.1.51.

Abstract

We constructed a soluble minimal receptor-Ig chimera in which the two extracellular domains of human Fcepsilonhain (D1 and D2) were fused to the dimerizing C-terminal domain of human IgG1 heavy chain (gamma1-CH3). The protein was expressed and actively secreted by Chinese hamster ovary (CHO) cells as a fully glycosylated soluble dimeric protein. It showed efficient binding both to human membrane-bound IgE isoforms and to the two secretory IgE isoforms. Moreover, the dimeric receptor binds IgE with the expected 1:2 stoichiometry. The receptor-Ig chimera, in 2-fold molar excess, inhibited engagement of secretory IgE to rat basophilic leukemia cells expressing the human alphabetagamma receptor. Full self-nature and inability to bind Fcgamma receptors make this protein an attractive candidate for clinical applications and a novel biotechnological tool for atopic allergy research.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • CHO Cells
  • Cell Line
  • Cricetinae
  • Dimerization
  • Humans
  • Immunoglobulin E / metabolism*
  • Immunoglobulin G / genetics
  • Membrane Proteins / metabolism
  • Mice
  • Models, Molecular
  • Protein Binding
  • Protein Isoforms / metabolism
  • Protein Structure, Tertiary
  • Protein Subunits
  • Rats
  • Receptors, IgE / chemistry
  • Receptors, IgE / genetics
  • Receptors, IgE / metabolism*
  • Recombinant Fusion Proteins / chemistry
  • Recombinant Fusion Proteins / metabolism
  • Solubility

Substances

  • Immunoglobulin G
  • Membrane Proteins
  • Protein Isoforms
  • Protein Subunits
  • Receptors, IgE
  • Recombinant Fusion Proteins
  • Immunoglobulin E