Abstract
Incubation of rat hippocampal slices with a low concentration of N-methyl-D-aspartate (NMDA; 20 microM; 3 min) elicits a form of long-term depression (LTD). We used this chemical protocol to study the involvement of pre- and postsynaptic protein kinase/phosphatase activity in NMDA receptor-dependent LTD. We determined the phosphorylation states of a pre- and a postsynaptic protein kinase C substrate, B-50/growth-associated protein 43 (GAP43) and RC3, respectively, using quantitative immunoprecipitation. NMDA incubation resulted in a 2-amino-5-phosphonovalerate-sensitive long-lasting (>60 min) decrease in synaptic efficacy and a concomitant reduction in RC3 phosphorylation. B-50/GAP43 phosphorylation was unaffected. This suggests that NMDA-LTD, in contrast to low frequency-LTD, is only associated with activation of postsynaptic protein phosphatases.
MeSH terms
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2-Amino-5-phosphonovalerate / pharmacology
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Animals
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Calmodulin-Binding Proteins / metabolism*
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Down-Regulation / drug effects
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Down-Regulation / physiology*
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Excitatory Amino Acid Antagonists / pharmacology
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Excitatory Postsynaptic Potentials / drug effects
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Excitatory Postsynaptic Potentials / physiology
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GAP-43 Protein / metabolism
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Hippocampus / cytology
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Hippocampus / drug effects
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Hippocampus / enzymology*
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Male
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N-Methylaspartate / pharmacology
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Nerve Tissue Proteins / metabolism*
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Neural Inhibition / drug effects
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Neural Inhibition / physiology*
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Neurogranin
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Neuronal Plasticity / drug effects
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Neuronal Plasticity / physiology*
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Phosphorylation / drug effects
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Protein Kinase C / antagonists & inhibitors
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Protein Kinase C / metabolism*
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Rats
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Rats, Wistar
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Receptors, N-Methyl-D-Aspartate / agonists
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Receptors, N-Methyl-D-Aspartate / metabolism*
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Synapses / drug effects
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Synapses / enzymology*
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Synaptic Transmission / drug effects
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Synaptic Transmission / physiology*
Substances
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Calmodulin-Binding Proteins
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Excitatory Amino Acid Antagonists
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GAP-43 Protein
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Nerve Tissue Proteins
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Nrgn protein, rat
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Receptors, N-Methyl-D-Aspartate
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Neurogranin
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N-Methylaspartate
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2-Amino-5-phosphonovalerate
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Protein Kinase C