Insulin-like growth factor binding protein-3 induces early apoptosis in malignant prostate cancer cells and inhibits tumor formation in vivo

Prostate. 2002 May 1;51(2):141-52. doi: 10.1002/pros.10068.

Abstract

Background: Insulin-like growth factor binding protein (IGFBP-3) levels are significantly reduced in malignant prostate epithelial cells. In this study, we evaluated the role of endogenous IGFBP-3 on prostate cancer cell growth and tumorigenesis.

Methods: IGFBP-3 was re-expressed by stable transfection of human IGFBP-3 cDNA in a model of human prostate cancer, M12, a malignant subline in which IGFBP-3 levels are undetectable in comparison to the parent epithelial cell, P69. Effect of IGFBP-3 re-expression (M12-BP-3) on growth kinetics, morphology, propensity to apoptosis, and in vivo tumor formation were studied.

Results: M12-BP-3 cells secreted IGFBP-3 and growth arrested at a cell density that was threefold lower than control cells and this was associated with marked alteration in cell morphology. Control cells when grown in conditioned media secreted by M12-BP-3 also showed altered morphology compared to when cultured in IGFBP-3-immunodepleted conditioned media. The M12-BP-3 clones showed altered mitochondrial membrane potential, increased PARP cleavage, increase in sub-G1 peak, decreased levels of neuron specific enolase, and decreased tumor formation in athymic, nude mice.

Conclusions: These data suggest that IGFBP-3 induces early apoptosis and has potential tumor suppressive effect in prostate cancer. Prostate 51: 141-152, 2002.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Apoptosis / drug effects*
  • Blotting, Western
  • Cell Division / drug effects*
  • Cell Transformation, Neoplastic*
  • Culture Media
  • DNA, Complementary / genetics
  • DNA, Neoplasm / genetics
  • Electrophoresis, Polyacrylamide Gel
  • Epithelial Cells / physiology
  • Gene Expression Regulation, Neoplastic*
  • Humans
  • Immunohistochemistry
  • Insulin-Like Growth Factor Binding Protein 3 / biosynthesis*
  • Insulin-Like Growth Factor Binding Protein 3 / pharmacology*
  • Male
  • Prostatic Neoplasms / pathology*
  • Tumor Cells, Cultured

Substances

  • Culture Media
  • DNA, Complementary
  • DNA, Neoplasm
  • Insulin-Like Growth Factor Binding Protein 3