Synthesis and anti-tubercular evaluation of 4-quinolylhydrazones

Bioorg Med Chem. 2002 Jul;10(7):2193-8. doi: 10.1016/s0968-0896(02)00071-8.

Abstract

A series of 4-quinolylhydrazones were synthesized and tested against Mycobacterium tuberculosis H37Rv. Preparation of the title compounds was achieved by reaction of 4-quinolylhydrazine and aryl- or heteroaryl-carboxaldehyde. For the most of derivatives interesting antitubercular properties were showed; two compounds (3(2) and 3(25)), identified as the most active, were tested also against Mycobacterium avium.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antitubercular Agents / chemical synthesis*
  • Antitubercular Agents / chemistry
  • Antitubercular Agents / pharmacology*
  • Drug Evaluation, Preclinical
  • Hydrazones / chemical synthesis*
  • Hydrazones / chemistry
  • Hydrazones / pharmacology*
  • Mycobacterium tuberculosis / drug effects

Substances

  • Antitubercular Agents
  • Hydrazones