Inhibition of glial glutamate transporter GLT-1 augments brain edema after transient focal cerebral ischemia in mice

Neurosci Lett. 2002 May 17;324(2):117-20. doi: 10.1016/s0304-3940(02)00193-3.

Abstract

Excessively released glutamate is neurotoxic. Glutamate transporters maintain the extracellular level of glutamate by uptake into glia or neurons. We examined the role of GLT-1, a glial glutamate transporter, in brain damage resulting from transient focal ischemia in mice. Heterozygous gene deletion of GLT-1 significantly augmented brain swelling resulting from 1 h of middle cerebral artery occlusion and 24 h reperfusion. In addition, this gene deletion significantly increased brain water contents in ischemic hemisphere at 6 h after reperfusion. Moreover, intraperitoneal injection of dihydrokainate (10 mg/kg), a specific inhibitor of GLT-1, augmented brain swelling. These data suggest that GLT-1 limits brain edema resulting from ischemia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain / drug effects
  • Brain / metabolism
  • Brain / physiopathology
  • Brain Edema / genetics*
  • Brain Edema / metabolism*
  • Brain Edema / physiopathology
  • Brain Ischemia / complications*
  • Excitatory Amino Acid Transporter 2 / antagonists & inhibitors
  • Excitatory Amino Acid Transporter 2 / deficiency*
  • Excitatory Amino Acid Transporter 2 / genetics
  • Extracellular Space / metabolism
  • Female
  • Glutamic Acid / metabolism*
  • Infarction, Middle Cerebral Artery / complications
  • Kainic Acid / analogs & derivatives*
  • Kainic Acid / pharmacology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Neuroglia / metabolism*
  • Neurotoxins / metabolism
  • Neurotransmitter Uptake Inhibitors / pharmacology
  • Reperfusion Injury / complications*
  • Water-Electrolyte Balance / genetics

Substances

  • Excitatory Amino Acid Transporter 2
  • Neurotoxins
  • Neurotransmitter Uptake Inhibitors
  • Glutamic Acid
  • dihydrokainic acid
  • Kainic Acid