Differential effect of gonadotropin-releasing hormone analogue treatment on estrogen levels and sulfatase activity in uterine leiomyoma and myometrium

Fertil Steril. 2002 Jun;77(6):1227-32. doi: 10.1016/s0015-0282(02)03093-5.

Abstract

Objective: To investigate the effect of GnRH treatment on estrogen levels and sulfatase activity in leiomyoma and myometrium tissue.

Design: Retrospective analyses of tissue obtained in a prospective randomized clinical study.

Setting: Gynecology departments of eight hospitals in the Netherlands.

Patient(s): Thirty-two patients scheduled for leiomyoma surgery.

Intervention(s): Patients were randomized to receive either GnRHa (3.75 mg/4 weeks of triptorelin or 3.6 mg/4 weeks of goserelin) or no GnRHa for 4 months. At subsequent surgery, leiomyoma and myometrium samples were collected.

Main outcome measure(s): Estrone, estradiol, and sulfatase activity levels in leiomyoma and myometrium.

Result(s): In myometrium, levels of estrone, estradiol, and sulfatase activity were significantly lower in the treated group (to median values of 46%, 21%, and 61%, respectively). In leiomyomas of treated patients, the reduction in median estrone level (to 65% of untreated value) was comparable to that in myometrium. The reduction in estradiol level in leiomyoma, however, was significantly less than in myometrium (median to 58% vs. 21%), and no significantly lower sulfatase activity was found.

Conclusion(s): Estradiol and sulfatase results show that the effect of GnRHa treatment on leiomyoma differs from the effect on myometrium, suggesting a continuing estrogenic stimulus in leiomyoma tissue despite treatment.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Antineoplastic Agents, Hormonal / therapeutic use*
  • Estradiol / metabolism*
  • Female
  • Goserelin / therapeutic use*
  • Humans
  • Leiomyoma / drug therapy
  • Leiomyoma / metabolism*
  • Myometrium / metabolism*
  • Randomized Controlled Trials as Topic
  • Retrospective Studies
  • Sulfatases / metabolism*
  • Triptorelin Pamoate / therapeutic use*
  • Uterine Neoplasms / drug therapy
  • Uterine Neoplasms / metabolism*

Substances

  • Antineoplastic Agents, Hormonal
  • Triptorelin Pamoate
  • Goserelin
  • Estradiol
  • Sulfatases
  • estrone sulfatase