The Fc receptor gamma-chain is necessary and sufficient to initiate signalling through glycoprotein VI in transfected cells by the snake C-type lectin, convulxin

Eur J Biochem. 2002 Jun;269(12):2951-60. doi: 10.1046/j.1432-1033.2002.02969.x.

Abstract

There is extensive evidence that FcR gamma-chain couples to the collagen receptor glycoprotein VI (GPVI) and becomes phosphorylated on tyrosines upon receptor cross-linking. However, it is not established whether this receptor complex is sufficient to initiate the signalling cascade. We transfected GPVI and the FcR gamma-chain into the human erythroleukaemia cell line K562, which lacks detectable expression of GPVI and the FcR gamma-chain. The results show that GPVI is unable to signal when expressed alone, despite its surface expression, upon stimulation with the snake C-type lectin, convulxin. Coexpression of the FcR gamma-chain confers signalling properties on the receptor. Furthermore, cotransfection of the FcR gamma-chain and two mutant versions of GPVI shows that the transmembrane arginine and cytoplasmic tail of GPVI are necessary for association with the FcR gamma-chain. These results demonstrate that reconstitution of the GPVI-FcR gamma-chain complex in cells expressing the necessary signalling network is sufficient to initiate signalling events in response to convulxin and collagen-related peptide.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arginine / metabolism
  • Binding Sites
  • COS Cells / metabolism
  • Calcium / metabolism
  • Carrier Proteins / pharmacology*
  • Chlorocebus aethiops
  • Collagen / pharmacology
  • Crotalid Venoms / genetics
  • Crotalid Venoms / pharmacology*
  • Enzyme Precursors / metabolism
  • Humans
  • Intracellular Signaling Peptides and Proteins
  • Jurkat Cells / metabolism
  • K562 Cells / drug effects
  • K562 Cells / metabolism
  • Lectins, C-Type*
  • Peptides*
  • Phosphorylation
  • Platelet Membrane Glycoproteins / metabolism*
  • Protein-Tyrosine Kinases / metabolism
  • Receptors, Fc / metabolism*
  • Signal Transduction / drug effects*
  • Signal Transduction / physiology
  • Syk Kinase
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Carrier Proteins
  • Crotalid Venoms
  • Enzyme Precursors
  • Intracellular Signaling Peptides and Proteins
  • Lectins, C-Type
  • Peptides
  • Platelet Membrane Glycoproteins
  • Receptors, Fc
  • collagen-related peptide
  • platelet membrane glycoprotein VI
  • convulxin
  • Collagen
  • Arginine
  • Protein-Tyrosine Kinases
  • SYK protein, human
  • Syk Kinase
  • Calcium