Protection of dopaminergic neurons in primary culture by lisuride

J Neural Transm (Vienna). 2002 Feb;109(2):157-69. doi: 10.1007/s007020200011.

Abstract

Dopamine agonists play an important role in the treatment of Parkinson's disease by reducing the administration of L-3,4-dihydroxyphenylalanine (L-DOPA). The enzymatic and non-enzymatic conversion of L-DOPA is suspected to increase oxidative stress, which leads to the degeneration of dopaminergic neurons in Parkinson's disease. In primary mouse mesencephalic cultures we show that the dopamine D1/D2 receptor agonist lisuride, in a concentration range of 0.001-1 microM, enhances the survival of dopaminergic neurons, protects against toxicity induced by L-DOPA or 1-methyl-4-phenylpyridinium ion (MPP+) and stimulates 3H-dopamine uptake. Lisuride also reduces anaerobic metabolism during incubation with L-DOPA. The present findings suggest that lisuride may have trophic/survival-promoting properties and potentially reduces oxidative stress.

MeSH terms

  • 1-Methyl-4-phenylpyridinium / toxicity
  • Animals
  • Antiparkinson Agents / pharmacology*
  • Antiparkinson Agents / toxicity
  • Cells, Cultured
  • Cytoprotection*
  • Dopamine / physiology*
  • Levodopa / toxicity
  • Lisuride / pharmacology*
  • Mesencephalon / drug effects
  • Mesencephalon / metabolism
  • Mice
  • Mice, Inbred C57BL
  • Neurons / drug effects*
  • Neurons / metabolism
  • Oxidative Stress / drug effects*

Substances

  • Antiparkinson Agents
  • Levodopa
  • Lisuride
  • 1-Methyl-4-phenylpyridinium
  • Dopamine