17beta-Estradiol upregulates distinct maxi-K channel transcripts in mouse uterus

Mol Cell Endocrinol. 2002 Jun 28;192(1-2):1-6. doi: 10.1016/s0303-7207(02)00136-3.

Abstract

The mouse maxi-K channel transcript undergoes alternative splicing to produce isoforms differing in sensitivity to intracellular regulators. We hypothesized that 17beta-estradiol could induce myometrial maxi-K channel transcripts to differentially splice. Polymerase chain reaction demonstrated two products at site D in mice injected with either 8.5 microg of 17beta-estradiol for 4 days or a vehicle control. Splicing of site D is known to modulate the sensitivity of the maxi-K channel to calcium and voltage. RNase protection analyses revealed that the alpha subunit transcript, and an exon encoding 59 amino acids at site D that enhances Ca(2+)- and voltage-sensitivity, are upregulated approximately 1.4-fold after 17beta-estradiol stimulation however, the insertless isoform of this transcript is enhanced approximately 5-fold. Immunoblotting demonstrates that the total maxi-K channel alpha subunit expression mimics transcript regulation. These findings verify that maxi-K channel transcripts are differentially spliced by 17beta-estradiol, which may contribute to stoichiometric changes in isoform expression during pregnancy.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alternative Splicing / drug effects*
  • Amino Acid Sequence
  • Animals
  • Base Sequence
  • Binding Sites
  • Calcium / metabolism
  • Estradiol / pharmacology*
  • Exons / genetics
  • Female
  • Large-Conductance Calcium-Activated Potassium Channel alpha Subunits
  • Large-Conductance Calcium-Activated Potassium Channels
  • Mice
  • Mice, Inbred C57BL
  • Models, Molecular
  • Molecular Sequence Data
  • Potassium Channels, Calcium-Activated / genetics*
  • Protein Subunits
  • Transcription, Genetic
  • Uterus / drug effects*
  • Uterus / metabolism

Substances

  • Large-Conductance Calcium-Activated Potassium Channel alpha Subunits
  • Large-Conductance Calcium-Activated Potassium Channels
  • Potassium Channels, Calcium-Activated
  • Protein Subunits
  • Estradiol
  • Calcium