Characterization of the interaction between murine tumour necrosis factor and monoclonal antibodies

Cytokine. 2002 May 7;18(3):158-63. doi: 10.1006/cyto.2002.0886.

Abstract

We characterized the interaction between murine TNF (mTNF) and the neutralizing monoclonal antibodies TN3 and 1F3F3. The epitopes were localized by comparing the detection efficiency for a panel of TNF chimaeric proteins and site-specific muteins in ELISA. Mutation of mTNF amino acid Q131 inhibited the interaction with 1F3F3, whereas mutation of D71/Y72 inhibited the binding to TN3. As D71/Y72 are located in an exposed loop near the TNF intersubunit groove, binding of TN3 promoted the dissociation and/or interfered with the reassociation of subunits into mTNF trimers. 1F3F3, on the other hand, prevented the spontaneous dissociation of bound (hetero)trimeric mTNF.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Monoclonal / metabolism*
  • Antigen-Antibody Reactions
  • Enzyme-Linked Immunosorbent Assay
  • Epitopes / chemistry
  • In Vitro Techniques
  • Kinetics
  • Mice
  • Models, Molecular
  • Mutagenesis, Site-Directed
  • Neutralization Tests
  • Protein Structure, Quaternary
  • Protein Subunits
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors
  • Tumor Necrosis Factor-alpha / chemistry
  • Tumor Necrosis Factor-alpha / genetics
  • Tumor Necrosis Factor-alpha / metabolism*

Substances

  • Antibodies, Monoclonal
  • Epitopes
  • Protein Subunits
  • Tumor Necrosis Factor-alpha