Synthesis and antioxidative properties of novel thiazolidinedione/imidazolidinedione compounds as retinoids

Pharmazie. 2002 Jul;57(7):438-41.

Abstract

The general term "retinoids" refers to both naturally occurring as well as synthetic compounds which exhibit biological activity similar to vitamin A (retinol). Vitamin A and its two metabolites, retinaldehyde and retinoic acid, are fat-soluble unsaturated isoprenoids necessary for the growth, differentiation and maintenance of epithelial tissues. In this study, we have synthesized thiazolidinedione/imidazolidinedione compounds as retinoids. Their in vitro effects on rat liver microsomal NADPH-dependent lipid peroxidation (LP) levels and superoxide anion formation were determined.

MeSH terms

  • Animals
  • Antioxidants / chemical synthesis*
  • Antioxidants / pharmacology*
  • Cytochrome c Group / chemistry
  • In Vitro Techniques
  • Indicators and Reagents
  • Lipid Peroxidation / drug effects
  • Male
  • Microsomes, Liver / drug effects
  • Microsomes, Liver / metabolism
  • NADP / metabolism
  • Rats
  • Retinoids / chemical synthesis*
  • Retinoids / pharmacology*
  • Superoxides / metabolism
  • Thiazoles / chemical synthesis*
  • Thiazoles / pharmacology*

Substances

  • Antioxidants
  • Cytochrome c Group
  • Indicators and Reagents
  • Retinoids
  • Thiazoles
  • Superoxides
  • NADP