Adenosine A2A analogue improves neurologic outcome after spinal cord trauma in the rabbit

J Trauma. 2002 Aug;53(2):225-9; discussion 229-31. doi: 10.1097/00005373-200208000-00005.

Abstract

Background: ATL-146e, an adenosine A2A agonist, reduces paralysis after spinal cord ischemia-reperfusion. We hypothesized that systemic ATL-146e could improve neurologic outcome after blunt spinal cord trauma.

Methods: Twenty rabbits survived a thoracic spinal cord impact of 30 g-cm. One group received 0.06 microg/kg/min ATL-146e for the first 3 hours after impact (A2A group), whereas a second group received saline carrier (T/C group). Neurologic outcome was measured using the Tarlov scale (0-5). Histologic sections from the A2A and T/C groups were compared for neuronal viability.

Results: There was significant improvement in Tarlov scores of A2A animals compared with T/C animals at 12 hours (p = 0.007), with a trend toward improvement at 36 (p = 0.08) and 48 (p = 0.09) hours after injury. There was decreased neuronal attrition in A2A animals (p = 0.06).

Conclusion: Systemic ATL-146e given after spinal cord trauma results in improved neurologic outcome. Adenosine A2A agonists may hold promise as a rapidly acting alternative to steroids in the early treatment of the spinal cord injured patient.

Publication types

  • Evaluation Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cyclohexanecarboxylic Acids / therapeutic use*
  • Hemodynamics / drug effects
  • Neuroprotective Agents / therapeutic use*
  • Paralysis / prevention & control*
  • Purinergic P1 Receptor Agonists*
  • Purines / therapeutic use*
  • Rabbits
  • Receptor, Adenosine A2A
  • Spinal Cord Injuries / drug therapy*
  • Spinal Cord Injuries / pathology
  • Spinal Cord Injuries / surgery
  • Statistics, Nonparametric
  • Wounds, Nonpenetrating / drug therapy*

Substances

  • ATL 146e
  • Cyclohexanecarboxylic Acids
  • Neuroprotective Agents
  • Purinergic P1 Receptor Agonists
  • Purines
  • Receptor, Adenosine A2A