Tumour Fas ligand:Fas ratio greater than 1 is an independent marker of relative resistance to tamoxifen therapy in hormone receptor positive breast cancer

Breast Cancer Res. 2002;4(5):R9. doi: 10.1186/bcr456. Epub 2002 Jun 21.

Abstract

Background: The objective of the present study was to examine the prognostic and predictive significance of the apoptosis-related marker Fas ligand (FasL):Fas ratio in breast cancer.

Methods: Tumour biopsies from 215 primary invasive breast cancer patients were examined for the expression of FasL and Fas mRNA transcripts by quantitative real-time RT-PCR. Their prognostic and predictive impact on patient survival was determined in univariate and multivariate survival analyses.

Results: Using a cutoff value of 1, a FasL:Fas ratio greater than 1 was found to have significant prognostic value for disease-free survival among the total population (median follow up 54 months). It was associated with a significantly decreased disease-free survival (P = 0.022) and with a tendency toward increased mortality (P = 0.14) in univariate analysis. Hormone receptor positive women exclusively treated with tamoxifen (n = 86) and with a FasL:Fas ratio greater than 1 had a significantly decreased disease-free survival (P = 0.008) and overall survival (P = 0.03) in univariate Kaplan-Meier analysis. Furthermore, tumour size and FasL:Fas ratio were of independent predictive significance in the multivariate model for disease-free and overall survival in that subgroup. Among postmenopausal patients (n = 148) both of those factors retained independent prognostic significance in the multivariate model for disease-free survival. In contrast, FasL:Fas ratio had no significant predictive value in patients exclusively treated with chemotherapy.

Conclusion: The data presented indicate that FasL:Fas ratio may be useful not only as a prognostic factor but also as a predictive factor for projecting response to the antioestrogen tamoxifen. The results strongly support a correlation between FasL:Fas ratio greater than 1 and lack of efficacy of tamoxifen in hormone receptor positive patients.

MeSH terms

  • Biomarkers, Tumor / genetics*
  • Biopsy
  • Breast Neoplasms / drug therapy
  • Breast Neoplasms / genetics*
  • Breast Neoplasms / mortality
  • Disease-Free Survival
  • Drug Resistance, Neoplasm / genetics*
  • Estrogen Antagonists / therapeutic use*
  • Fas Ligand Protein
  • Female
  • Humans
  • Ligands
  • Membrane Glycoproteins / genetics*
  • Membrane Glycoproteins / metabolism
  • Neoplasm Invasiveness / pathology
  • Neoplasms, Hormone-Dependent / drug therapy
  • Neoplasms, Hormone-Dependent / genetics*
  • Neoplasms, Hormone-Dependent / mortality
  • Prognosis
  • RNA, Messenger / metabolism
  • Receptors, Estrogen / metabolism
  • Receptors, Progesterone / metabolism
  • Reverse Transcriptase Polymerase Chain Reaction
  • Survival Rate
  • Tamoxifen / therapeutic use*
  • fas Receptor / genetics*
  • fas Receptor / metabolism

Substances

  • Biomarkers, Tumor
  • Estrogen Antagonists
  • FASLG protein, human
  • Fas Ligand Protein
  • Ligands
  • Membrane Glycoproteins
  • RNA, Messenger
  • Receptors, Estrogen
  • Receptors, Progesterone
  • fas Receptor
  • Tamoxifen