Non-Fc-mediated mechanisms are involved in clearance of amyloid-beta in vivo by immunotherapy

J Neurosci. 2002 Sep 15;22(18):7873-8. doi: 10.1523/JNEUROSCI.22-18-07873.2002.

Abstract

Transgenic (Tg) mouse models overexpressing amyloid precursor protein (APP) develop senile plaques similar to those found in Alzheimer's disease in an age-dependent manner. Recent reports demonstrated that immunotherapy is effective at preventing or removing amyloid-beta deposits in the mouse models. To characterize the mechanisms involved in clearance, we used antibodies of either IgG1 (10d5) or IgG2b (3d6) applied directly to the brains of 18-month-old Tg2576 or 20-month-old PDAPP mice. Both 10d5 and 3d6 led to clearance of 50% of diffuse amyloid deposits in both animal models within 3 d. Fc receptor-mediated clearance has been shown to be important in an ex vivo assay showing antibody-mediated clearance of plaques by microglia. We now show, using in vivo multiphoton microscopy, that FITC-labeled F(ab')2 fragments of 3d6 (which lack the Fc region of the antibody) also led to clearance of 45% of the deposits within 3 d, similar to the results obtained with full-length 3d6 antibody. This result suggests that direct disruption of plaques, in addition to Fc-dependent phagocytosis, is involved in the antibody-mediated clearance of amyloid-beta deposits in vivo. Dense-core deposits that were not cleared were reduced in size by approximately 30% with full-length antibodies and F(ab')2 fragments 3 d after a topical treatment. Together, these results indicate that clearance of amyloid deposits in vivo may involve, in addition to Fc-dependent clearance, a non-Fc-mediated disruption of plaque structure.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Administration, Topical
  • Alzheimer Disease / immunology
  • Alzheimer Disease / metabolism*
  • Alzheimer Disease / pathology
  • Alzheimer Disease / therapy
  • Amyloid beta-Peptides / immunology
  • Amyloid beta-Peptides / metabolism*
  • Amyloid beta-Protein Precursor / genetics
  • Amyloid beta-Protein Precursor / metabolism
  • Animals
  • Antibodies / administration & dosage
  • Benzothiazoles
  • Brain / metabolism
  • Brain / pathology
  • Disease Models, Animal
  • Fluorescent Dyes
  • Humans
  • Immunoglobulin Fab Fragments / pharmacology
  • Immunoglobulin Fc Fragments / metabolism*
  • Immunotherapy*
  • Mice
  • Mice, Transgenic
  • Microscopy, Fluorescence / methods
  • Mutation
  • Phagocytosis / immunology
  • Plaque, Amyloid / drug effects
  • Plaque, Amyloid / metabolism
  • Thiazoles

Substances

  • Amyloid beta-Peptides
  • Amyloid beta-Protein Precursor
  • Antibodies
  • Benzothiazoles
  • Fluorescent Dyes
  • Immunoglobulin Fab Fragments
  • Immunoglobulin Fc Fragments
  • Thiazoles
  • thioflavin T