Intrahippocampal infusion of ebselen impairs retention of an inhibitory avoidance task in rats

Eur J Pharmacol. 2002 Sep 13;451(2):165-9. doi: 10.1016/s0014-2999(02)02221-5.

Abstract

Ebselen is a seleno-compound used in the treatment of neurological disorders involving the glutamatergic system. Although ebselen is currently used in clinical trials, the physiological effects of this seleno-compound are poorly known. In this study, we investigated the effects of intrahippocampal infusion of ebselen (0.1-3 nmol) in rats submitted to an inhibitory avoidance task. Ebselen (1-3 nmol) infused after the training session impaired retention of inhibitory avoidance, tested 90 min or 24 h after the training session. Moreover, ebselen also impaired the retention when infused 30 min prior to training or 10 min prior to test sessions. In summary, ebselen impaired memory consolidation, acquisition and retrieval. This amnesic effect of ebselen could be related to oxidant activity at N-methyl-D-aspartate (NMDA) receptors. Our results indicate that more studies must be performed to investigate the mechanisms of this amnesic effect and whether ebselen has a cognition-impairing effect when administered chronically.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Avoidance Learning / drug effects*
  • Avoidance Learning / physiology
  • Azoles / administration & dosage*
  • Dose-Response Relationship, Drug
  • Hippocampus / drug effects*
  • Hippocampus / physiology
  • Infusion Pumps
  • Isoindoles
  • Male
  • Motor Activity / drug effects
  • Motor Activity / physiology
  • Organoselenium Compounds / administration & dosage*
  • Rats
  • Rats, Wistar
  • Retention, Psychology / drug effects*
  • Retention, Psychology / physiology

Substances

  • Azoles
  • Isoindoles
  • Organoselenium Compounds
  • ebselen