Role of endothelin B receptor in the pathogenesis of ischemic acute renal failure

J Cardiovasc Pharmacol. 2002 Oct;40(4):586-93. doi: 10.1097/00005344-200210000-00012.

Abstract

This study evaluated the role of endothelin B (ET ) receptor-mediated action in the development and maintenance of ischemic acute renal failure (ARF), using the spotting-lethal ( ) rat that carries a naturally occurring deletion in the ET receptor gene. Because homozygous ( ) rats die shortly after birth due to congenital distal intestinal aganglionosis, genetic rescue of rats from the developmental defect using a dopamine-beta-hydroxylase (DbetaH)-ET transgene was performed to produce ET -deficient adult rats. Rescued homozygous (DbetaH-ET ) and wild-type (DbetaH-ET +/+) rats were subjected to ischemic ARF by clamping the renal pedicle for 45 min followed by reperfusion. At 24 h after the reperfusion, renal glomerular dysfunction and histologic damage, such as proteinaceous casts in tubuli, were markedly and observed equally in homozygous and wild-type groups, and these renal injuries gradually recovered. However, when the ischemia/reperfusion-induced renal injury was examined 7 days after the reperfusion, the recovery in homozygous ARF rats was obviously delayed compared with the wild-type animals. Two of the eight homozygous ARF rats died within 3 days after the reperfusion. Increment of renal endothelin-1 content after the ischemia/reperfusion was more marked in homozygous than in wild-type rats. Thus, ET receptor-mediated actions do not play an important role in the development of ischemic ARF but may be involved in the recovery process from ischemia/reperfusion-induced renal injury.

Publication types

  • Comparative Study

MeSH terms

  • Acute Kidney Injury / genetics
  • Acute Kidney Injury / pathology
  • Acute Kidney Injury / physiopathology*
  • Animals
  • Animals, Genetically Modified
  • Endothelin-1 / metabolism
  • Ischemia / genetics
  • Ischemia / pathology
  • Ischemia / physiopathology*
  • Kidney / blood supply
  • Kidney / pathology
  • Rats
  • Receptor, Endothelin B
  • Receptors, Endothelin / deficiency
  • Receptors, Endothelin / genetics
  • Receptors, Endothelin / physiology*

Substances

  • Endothelin-1
  • Receptor, Endothelin B
  • Receptors, Endothelin