DAP-kinase induces apoptosis by suppressing integrin activity and disrupting matrix survival signals

J Cell Biol. 2002 Oct 14;159(1):169-79. doi: 10.1083/jcb.200204050. Epub 2002 Oct 7.

Abstract

Death-associated protein kinase (DAP-kinase) is a calcium/calmodulin-dependent serine/threonine kinase, and participates in various apoptosis systems. However, its apoptosis-promoting mechanism is poorly understood. Here, we demonstrate that DAP-kinase suppresses integrin-mediated cell adhesion and signal transduction, whereas dominant-negative interference of this kinase promotes adhesion. This effect of DAP-kinase is neither a consequence of apoptosis nor a result of decreased expression of integrins. Rather, DAP-kinase downregulates integrin activity through an inside-out mechanism. We present evidence indicating that this adhesion-inhibitory effect accounts for a major mechanism of the apoptosis induced by DAP-kinase. First, in growth-arrested fibroblasts, DAP-kinase triggers apoptosis in cells plated on fibronectin, but does not affect the death of cells on poly-l-lysine. Second, in epithelial cells, DAP-kinase induces apoptosis in the anoikis-sensitive MCF10A cells, but not in the anoikis-resistant BT474 cells. Most importantly, the apoptosis-promoting effect of DAP-kinase is completely abolished by enforced activation of integrin-mediated signaling pathways from either integrin itself or its downstream effector, FAK. Finally, we show that integrin or FAK activation blocks the ability of DAP-kinase to upregulate p53. Our results indicate that DAP-kinase exerts apoptotic effects by suppressing integrin functions and integrin-mediated survival signals, thereby activating a p53-dependent apoptotic pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Chloromethyl Ketones / metabolism
  • Animals
  • Apoptosis / physiology*
  • Apoptosis Regulatory Proteins
  • Breast Neoplasms / metabolism
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
  • Carcinoma / metabolism
  • Caspase 3
  • Caspase Inhibitors
  • Caspases / metabolism
  • Cell Adhesion / physiology*
  • Cell Line
  • Cell Size
  • Cell Survival
  • Cysteine Proteinase Inhibitors / metabolism
  • Death-Associated Protein Kinases
  • Epithelial Cells / cytology
  • Epithelial Cells / metabolism
  • Extracellular Matrix / metabolism*
  • Genes, Reporter
  • Humans
  • Integrins / metabolism*
  • Mice
  • Signal Transduction / physiology*
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / metabolism

Substances

  • Amino Acid Chloromethyl Ketones
  • Apoptosis Regulatory Proteins
  • Caspase Inhibitors
  • Cysteine Proteinase Inhibitors
  • Integrins
  • Tumor Suppressor Protein p53
  • benzyloxycarbonylvalyl-alanyl-aspartyl fluoromethyl ketone
  • Death-Associated Protein Kinases
  • Calcium-Calmodulin-Dependent Protein Kinases
  • CASP3 protein, human
  • Casp3 protein, mouse
  • Caspase 3
  • Caspases