Effects of slow-release octreotide on urinary metanephrine excretion and plasma chromogranin A and catecholamine levels in patients with malignant or recurrent phaeochromocytoma

Clin Endocrinol (Oxf). 2002 Nov;57(5):629-34. doi: 10.1046/j.1365-2265.2002.01658.x.

Abstract

Objective: Somatostatin receptors are present on human phaeochromocytomas. Catecholamine concentrations may decrease following short-term administration of somatostatin agonists to patients with phaeochromocytomas. We carried out a prospective study on 10 patients with malignant or recurrent phaeochromocytomas to examine the clinical and hormonal effects of three monthly intramuscular injections of 20 mg slow-release octreotide.

Design and measurements: Patients underwent somatostatin receptor scintigraphy using 111In-pentetreotide before slow-release octreotide was administered. The patients' symptoms, blood pressure, blood glucose concentrations, glycosylated haemoglobin concentra-tions, plasma insulin and noradrenaline concentrations, and the levels of two putative markers of tumour burden, urinary metanephrine excretion and plasma chromogranin A concentration, were recorded before the first injection and 28 days after the third injection.

Results: Slow-release octreotide did not significantly alter symptoms, blood pressure, blood glucose concentrations, plasma catecholamine and chromogranin A concentrations or metanephrine excretion. Median glycosylated haemoglobin concentrations increased from 5.3% to 6.0% (P = 0.03). Patients whose tumours took up 111In- pentetreotide did not differ from those whose tumours did not after slow-release octreotide treatment in terms of symptoms, blood pressure, blood glucose, plasma catecholamine and chromogranin A concentrations or metanephrine excretion.

Conclusion: Our data suggest that slow-release octreotide is of limited value for the long-term treatment of patients with malignant or recurrent benign phaeochromocytomas.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenal Gland Neoplasms* / blood
  • Adrenal Gland Neoplasms* / drug therapy
  • Adrenal Gland Neoplasms* / urine
  • Adult
  • Aged
  • Biomarkers, Tumor* / blood
  • Biomarkers, Tumor* / urine
  • Blood Pressure
  • Catecholamines / urine*
  • Chromogranin A
  • Chromogranins / blood*
  • Delayed-Action Preparations
  • Female
  • Heart Rate
  • Humans
  • Injections, Intramuscular
  • Male
  • Metanephrine / urine*
  • Middle Aged
  • Octreotide / administration & dosage*
  • Octreotide / therapeutic use
  • Pheochromocytoma* / blood
  • Pheochromocytoma* / drug therapy
  • Pheochromocytoma* / urine
  • Prospective Studies
  • Somatostatin / analogs & derivatives*
  • Somatostatin / pharmacokinetics

Substances

  • Biomarkers, Tumor
  • CHGA protein, human
  • Catecholamines
  • Chromogranin A
  • Chromogranins
  • Delayed-Action Preparations
  • Metanephrine
  • Somatostatin
  • pentetreotide
  • Octreotide