Impairment of male fertility induced by muscarinic receptor antagonists in rats

Reprod Toxicol. 2002 Nov-Dec;16(6):757-65. doi: 10.1016/s0890-6238(02)00050-3.

Abstract

Male rats were treated with a muscarinic receptor antagonist at 3, 10, and 100mg/kg/day for 4 weeks prior to mating with untreated females and their reproductive status was determined on gestation days (GD) 15-17. Treatment-related decreases in the pregnancy rate were observed at 100mg/kg/day without any effects on mating performance. Impairment of male fertility by this compound was also observed after treatment for 1 week, but there were no effects after a 1-week withdrawal period suggesting reversibility of the effect. There were no treatment-related effects on sperm production or motility, or testicular histopathology in any group. In order to determine whether the reduced fertility was a class effect of muscarinic receptor antagonists, atropine was examined. Males received atropine for 1 week at 62.5 and 125 mg/kg/day and were mated with untreated females. A low pregnancy rate associated with a decrease in the number of implantations was observed at 125 mg/kg/day. The effect on implantation was also observed at 62.5mg/kg/day. These findings suggest that the impairment of fertility in male rats induced by muscarinic receptor antagonists is a class effect, and has a relatively short onset of effect and is quickly reversible.

MeSH terms

  • Administration, Oral
  • Animals
  • Atropine / administration & dosage
  • Atropine / toxicity*
  • Dose-Response Relationship, Drug
  • Drug Evaluation, Preclinical
  • Female
  • Fertility / drug effects*
  • Fertility / physiology
  • Male
  • Muscarinic Antagonists / administration & dosage
  • Muscarinic Antagonists / toxicity*
  • Pregnancy
  • Pregnancy Rate
  • Rats
  • Rats, Inbred Strains
  • Recovery of Function
  • Spermatogenesis / drug effects*
  • Spermatogenesis / physiology

Substances

  • Muscarinic Antagonists
  • Atropine