Orexin-mediated feeding behavior involves both leptin-sensitive and -insensitive pathways

Physiol Behav. 2002 Nov;77(2-3):251-7. doi: 10.1016/s0031-9384(02)00843-0.

Abstract

Orexin-A and -B are neuropeptides that are implicated in the regulation of vigilance states and energy homeostasis. Orexins are specifically produced by neurons located within the lateral hypothalamic area (LHA), a region implicated in the regulation of feeding behavior. Here, we examined the functional interactions between orexins and anorectic factors [leptin, alpha-melanocyte-stimulating hormone (alpha-MSH) and glucagon-like peptide-1 (GLP-1)] in rats. Intracerebroventricular injection of orexin-A (10 nmol) potently augmented food intake in rats. Neuropeptide Y (NPY) (0.3 nmol) and galanin (3 nmol) also induced a transient increase in food intake. Both NPY- and galanin-induced feeding behaviors were completely inhibited by preadministration of leptin (3 microg), while the same or a higher dose (10 microg) of leptin only partially inhibited orexin-A or -B-induced increase of food intake. Preadministration of anorectic peptides (alpha-MSH and GLP-1), which are shown to be regulated by leptin, abolished NPY-induced feeding; however, orexin-induced feeding was only partially inhibited by these anorectic peptides. These observations suggest that NPY- and galanin-induced increases of feeding involve a leptin-sensitive pathway, while orexin-induced feeding involves both leptin-sensitive and -insensitive pathways.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Carrier Proteins / pharmacology*
  • Feeding Behavior / drug effects*
  • Galanin / pharmacology
  • Glucagon / pharmacology
  • Glucagon-Like Peptide 1
  • Injections, Intraventricular
  • Intracellular Signaling Peptides and Proteins*
  • Leptin / pharmacology*
  • Male
  • Neuropeptides / pharmacology*
  • Orexin Receptors
  • Orexins
  • Peptide Fragments / pharmacology
  • Protein Precursors / pharmacology
  • Rats
  • Rats, Wistar
  • Receptors, G-Protein-Coupled
  • Receptors, Neuropeptide
  • Receptors, Neuropeptide Y / antagonists & inhibitors
  • alpha-MSH / pharmacology

Substances

  • Carrier Proteins
  • Intracellular Signaling Peptides and Proteins
  • Leptin
  • Neuropeptides
  • Orexin Receptors
  • Orexins
  • Peptide Fragments
  • Protein Precursors
  • Receptors, G-Protein-Coupled
  • Receptors, Neuropeptide
  • Receptors, Neuropeptide Y
  • neuropeptide Y-Y1 receptor
  • alpha-MSH
  • Galanin
  • Glucagon-Like Peptide 1
  • Glucagon