Platelet factor 4 enhances the binding of oxidized low-density lipoprotein to vascular wall cells

J Biol Chem. 2003 Feb 21;278(8):6187-93. doi: 10.1074/jbc.M208894200. Epub 2002 Dec 3.

Abstract

Accumulation of low-density lipoprotein (LDL)-derived cholesterol by macrophages in vessel walls is a pathogenomic feature of atherosclerotic lesions. Platelets contribute to lipid uptake by macrophages through mechanisms that are only partially understood. We have previously shown that platelet factor 4 (PF4) inhibits the binding and degradation of LDL through its receptor, a process that could promote the formation of oxidized LDL (ox-LDL). We have now characterized the effect of PF4 on the binding of ox-LDL to vascular cells and macrophages and on the accumulation of cholesterol esters. PF4 bound to ox-LDL directly and also increased ox-LDL binding to vascular cells and macrophages. PF4 did not stimulate ox-LDL binding to cells that do not synthesize glycosaminoglycans or after enzymatic cleavage of cell surface heparan and chondroitin sulfates. The effect of PF4 on binding ox-LDL was dependent on specific lysine residues in its C terminus. Addition of PF4 also caused an approximately 10-fold increase in the amount of ox-LDL esterified by macrophages. Furthermore, PF4 and ox-LDL co-localize in atherosclerotic lesion, especially in macrophage-derived foam cells. These observations offer a potential mechanism by which platelet activation at sites of vascular injury may promote the accumulation of deleterious lipoproteins and offer a new focus for pharmacological intervention in the development of atherosclerosis.

MeSH terms

  • Amino Acid Substitution
  • Animals
  • Arteriosclerosis / pathology
  • Blood Platelets / physiology*
  • CHO Cells
  • Cells, Cultured
  • Cricetinae
  • Endothelium, Vascular / pathology
  • Endothelium, Vascular / physiology*
  • Genetic Variation
  • Humans
  • Immunohistochemistry
  • Lipoproteins, LDL / metabolism*
  • Microscopy, Confocal
  • Mutagenesis, Site-Directed
  • Platelet Factor 4 / chemistry
  • Platelet Factor 4 / genetics
  • Platelet Factor 4 / pharmacology*
  • Protein Binding
  • Proteoglycans / pharmacology
  • Recombinant Proteins / metabolism
  • Transfection
  • Umbilical Veins

Substances

  • Lipoproteins, LDL
  • Proteoglycans
  • Recombinant Proteins
  • oxidized low density lipoprotein
  • Platelet Factor 4