[A humanized anti-IL-6 receptor antibody(MRA) in RA therapy]

Nihon Rinsho. 2002 Dec;60(12):2401-7.
[Article in Japanese]

Abstract

Hyperproduction of Interleukin-6(IL-6) is observed in the rheumatoid arthritis(RA) patients and serum level of IL-6 is closely related to disease activity. IL-6 is a pleiotropic cytokine and its hyperfunctions explain most of the clinical symptoms in RA. Since MRA is humanized antibody from a mouse anti-human IL-6 receptor antibody, MRA can be administered repeatedly because of its low antigenesity to human. MRA inhibits IL-6 function by the blocking IL-6 binding to IL-6 receptor, resulting the prevention of development on collagen inducing arthritis(CIA) in cynomolgus monkeys whose IL-6R is cross-reacted with MRA. These evidence suggest that MRA has anti-arthritic effects. Clinical trials of MRA for RA patients have already started, and MRA therapy is effective as well as anti-TNF alpha and anti-IL-1 therapies.

Publication types

  • English Abstract
  • Review

MeSH terms

  • Animals
  • Antibodies, Monoclonal / therapeutic use*
  • Arthritis, Rheumatoid / drug therapy*
  • Humans
  • Interleukin-6 / physiology
  • Mice
  • Receptors, Interleukin-6 / chemistry
  • Receptors, Interleukin-6 / immunology*
  • Signal Transduction

Substances

  • Antibodies, Monoclonal
  • Interleukin-6
  • Receptors, Interleukin-6