Coronary flow-induced inotropism is modulated by binding of dextrans to the endothelial luminal surface

Am J Physiol Heart Circ Physiol. 2003 Apr;284(4):H1348-57. doi: 10.1152/ajpheart.00323.2002. Epub 2003 Jan 2.

Abstract

In isolated perfused guinea pig hearts, coronary flow causes a positive inotropic effect [positive coronary flow-induced effect (+CFIE)] that could be altered by dextrans (Dx) in the coronary perfusion solution. To test this possibility, Dx of 20, 40, 70, and 500 kDa were infused and found to modulate +CFIE; however, when Dx infusion was terminated, the effect persisted, i.e., was irreversible/nonwashable, suggesting that Dx may bind to luminal endothelial lectinic structures. This hypothesis was tested when Dx [with fluorescent traces (D*)] bound to the vessel wall was hydrolyzed by dextranase infusion and washout of D* fragments completely reverted the +CFIE, and it was found that bound D* to be displaced by free Dx required concentrations 50-100 times that used during binding. In addition, dose-response curves for Dx on +CFIE show that the higher the Dx molecular mass, the lesser the concentration required to have an effect. Because a large Dx molecule has a greater number polymeric glucose branches, it can bind to a larger number of endothelial lectinic sites, requiring a lower concentration to affect +CFIE. Our results suggest that luminal endothelial lectinic structures are part of the flow-sensing assembly.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Albumins / administration & dosage
  • Albumins / metabolism
  • Animals
  • Blood Flow Velocity
  • Coronary Circulation*
  • Dextrans / administration & dosage*
  • Dextrans / chemistry
  • Dextrans / metabolism*
  • Endothelium, Vascular / metabolism*
  • Fluorescein-5-isothiocyanate / administration & dosage
  • Fluorescein-5-isothiocyanate / analogs & derivatives*
  • Fluorescein-5-isothiocyanate / metabolism
  • Fluorescent Dyes
  • Guinea Pigs
  • Kinetics
  • Male
  • Molecular Weight
  • Muscle Contraction / drug effects
  • Muscle Contraction / physiology*
  • Solutions
  • Stimulation, Chemical
  • Viscosity

Substances

  • Albumins
  • Dextrans
  • Fluorescent Dyes
  • Solutions
  • fluorescein isothiocyanate dextran
  • Fluorescein-5-isothiocyanate