Mechanism of inhibition of RNA polymerase I transcription by DNA-dependent protein kinase

Biol Chem. 2002 Nov;383(11):1683-90. doi: 10.1515/BC.2002.189.

Abstract

DNA-dependent protein kinase represses RNA polymerase I (Pol I) transcription in vitro. To investigate the mechanism underlying transcriptional repression, we compared Pol I transcription in extracts from cells that either contain or lack the catalytic subunit of DNA-PK (DNA-PKcs). ATP-dependent repression of Pol I transcription was observed in extracts from DNA-PKcs-containing but not -deficient cells, required templates with free DNA ends, and was overcome by exogenous SL1, the factor that nucleates initiation complex formation. Order-of-addition experiments demonstrate that DNA-PKcs does not inactivate component(s) of the Poll transcription machinery. Instead, phosphorylated Ku protein competes with SL1 for binding to the rDNA promoter and, as a consequence, prevents initiation complex formation. The results reveal a novel mechanism of transcriptional regulation by DNA-PK. Once targeted to DNA, autophosphorylated Ku may displace positive- or negative-acting factors from their target sites, thereby repressing or activating transcription in a gene-specific manner.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antigens, Nuclear / metabolism
  • Blotting, Western
  • DNA / physiology*
  • DNA Helicases*
  • DNA, Ribosomal / biosynthesis
  • DNA-Binding Proteins / metabolism
  • Electrophoretic Mobility Shift Assay
  • Enzyme Inhibitors / pharmacology
  • Humans
  • Ku Autoantigen
  • Phosphoric Monoester Hydrolases / antagonists & inhibitors
  • Phosphorylation
  • Pol1 Transcription Initiation Complex Proteins / physiology
  • Promoter Regions, Genetic / drug effects
  • Protein Kinases / pharmacology*
  • RNA Polymerase I / antagonists & inhibitors*
  • RNA Polymerase I / biosynthesis*
  • Transcription, Genetic / drug effects*
  • Tumor Cells, Cultured

Substances

  • Antigens, Nuclear
  • DNA, Ribosomal
  • DNA-Binding Proteins
  • Enzyme Inhibitors
  • Pol1 Transcription Initiation Complex Proteins
  • transcription initiation factor TIF-IB
  • DNA
  • Protein Kinases
  • RNA Polymerase I
  • Phosphoric Monoester Hydrolases
  • DNA Helicases
  • XRCC5 protein, human
  • Xrcc6 protein, human
  • Ku Autoantigen