Absence of thermal hyperalgesia in serotonin transporter-deficient mice

J Neurosci. 2003 Jan 15;23(2):708-15. doi: 10.1523/JNEUROSCI.23-02-00708.2003.

Abstract

Antidepressants in the treatment of neuropathic pain are thought to partially exert their effect by inhibition of serotonin (5-HT) reuptake and thus activation of central antinociceptive pathways. Mice deficient for the 5-HT transporter (5-HTT-/- mice) are regarded as a model of lifelong treatment with a serotonin reuptake inhibitor. Here we investigated 5-HTT-/- mice and compared their pain-related behavior after a unilateral chronic constrictive sciatic nerve injury (CCI) with that of wild-type littermates. Wild-type mice reproducibly developed ipsilateral thermal hyperalgesia and mechanical allodynia after CCI. 5-HTT-/- mice did not develop thermal hyperalgesia, but showed bilateral mechanical allodynia after the nerve injury. 5-HT levels as measured with HPLC increased after CCI in the injured nerve in both genotypes and decreased in the lumbar spinal cord in wild-type mice. 5-HTT-/- mice had significantly lower 5-HT concentrations than wild-type mice in all tissues investigated. Thus, in 5-HTT-/- mice, reduced 5-HT levels in the injured peripheral nerves correlate with diminished behavioral signs of thermal hyperalgesia, a pain-related symptom caused by peripheral sensitization. In contrast, bilateral mechanical allodynia, a centrally mediated phenomenon, was associated with decreased spinal 5-HT concentrations in 5-HTT-/- mice and may possibly be caused by a lack of spinal inhibition.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenal Glands / metabolism
  • Animals
  • Behavior, Animal
  • Carrier Proteins / genetics
  • Disease Models, Animal
  • Hindlimb / physiopathology
  • Hot Temperature
  • Hydroxyindoleacetic Acid / metabolism
  • Hyperalgesia / physiopathology*
  • Lumbosacral Region
  • Membrane Glycoproteins / deficiency*
  • Membrane Glycoproteins / genetics
  • Membrane Transport Proteins*
  • Mice
  • Mice, Knockout
  • Nerve Tissue Proteins*
  • Pain Measurement
  • Pain Threshold
  • Reaction Time
  • Sciatic Nerve / physiopathology
  • Sciatic Neuropathy / physiopathology*
  • Serotonin / metabolism
  • Serotonin Plasma Membrane Transport Proteins
  • Skin Temperature
  • Spinal Cord / physiopathology

Substances

  • Carrier Proteins
  • Membrane Glycoproteins
  • Membrane Transport Proteins
  • Nerve Tissue Proteins
  • Serotonin Plasma Membrane Transport Proteins
  • Slc6a4 protein, mouse
  • Serotonin
  • Hydroxyindoleacetic Acid