Chorion-induced myometrial relaxation is mediated by large-conductance Ca2+-activated K+ channel opening in the guinea pig

Am J Obstet Gynecol. 2003 Jan;188(1):84-91. doi: 10.1067/mob.2003.102.

Abstract

Objective: We previously demonstrated that chorion releases a factor that inhibits both spontaneous and oxytocin-stimulated myometrial contractility. Here, we investigate the mechanism of action of this unidentified substance.

Study design: Myometrial strips from pregnant guinea pigs were mounted in an organ bath and contractility stimulated with oxytocin.

Results: Guinea pig chorion produced a time-dependent decrease in oxytocin-induced myometrial contractility. The ability of the chorion to reduce contractility was unaltered by inhibiting chorionic synthesis of either nitric oxide (N [omega]-nitro-L-arginine), carbon monoxide (tin-protoporphyrin), prostaglandins (indomethacin), or the myometrial cyclic guanosine monophosphate pathway (1H-[1,2,4]oxadiazolo[4,3-a]quinoxalime-1-one and Rp-8Br-cGMP). In contrast, iberiotoxin, an inhibitor of large conductance Ca(2+)-activated K(+) channels reduced the quiescent effect of chorion by 40%; in contrast, inhibition of adenosine triphosphate-sensitive (glibenclamide) and voltage-gated K(+) channels (4amynopyridine) had no effect.

Conclusion: Chorion-induced relaxation of oxytocin-stimulated myometrial contraction is, in great part, the product of a paracrine substance that opens myometrial large conductance Ca(2+)-activated K(+) channels.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Chorion / physiology*
  • Culture Media, Conditioned
  • Culture Techniques
  • Cyclic GMP / analogs & derivatives*
  • Cyclic GMP / pharmacology
  • Cyclic GMP / physiology
  • Cyclic GMP-Dependent Protein Kinases / antagonists & inhibitors
  • Cyclic GMP-Dependent Protein Kinases / metabolism
  • Enzyme Inhibitors / pharmacology
  • Female
  • Guinea Pigs
  • Ion Channel Gating / physiology*
  • Muscle Relaxation*
  • Myometrium / physiology*
  • Peptides / pharmacology
  • Potassium Channel Blockers / pharmacology
  • Potassium Channels, Calcium-Activated / physiology*
  • Pregnancy
  • Tetraethylammonium / pharmacology
  • Thionucleotides
  • Uterine Contraction

Substances

  • Culture Media, Conditioned
  • Enzyme Inhibitors
  • Peptides
  • Potassium Channel Blockers
  • Potassium Channels, Calcium-Activated
  • Thionucleotides
  • 8-bromoguanosino-3',5'-cyclic monophosphorothioate
  • Tetraethylammonium
  • iberiotoxin
  • Cyclic GMP-Dependent Protein Kinases
  • Cyclic GMP