[The study on Rhizoma Alpiniae officinarum and other herbs as penetration enhancer for the permeation of 5-fluorouacil]

Zhong Yao Cai. 2000 Nov;23(11):697-9.
[Article in Chinese]

Abstract

Objective: To study the effects of volatile oils from Rhizoma Alpiniae Officinarum, Pericarpium Zanthoxyli, Herba Asari, cineaol and ethanol extracts on the percutaneous pentration of 5-fluorouracil.

Methods: By Valia-Chienhorizontal diffusion cell and HPLC, the effects of volatile oils from Rhizoma Alpiniae Officinarum, Pericarpium Zanthoxyli, Herba Asari, cineol and ethanol extracts on the percutaneous penetration of 5-fluorouracil were observed and compared with azone.

Result: 1%, 3% volatile oils from Rhizoma Alpiniae Officinarum, Pericarpium Zanthoxyli and cineol possessed strong promoting action on percutaneous absorption of 5-fluorouracil. The effects of volatile oils from Rhizoma Alpiniae Officinarum was stronger than that of azone; the effects of volatile oils from Pericarpium Zanthoxyli was the same as that of azone. CONDUSION: The volatile oils from Rhizoma Alpiniae Officinarum, Pericarpium Zanthoxyli, Herba Asari can enhance effectively the skin permeation of 5-fluorouracil. They deserved to be researched and developed further.

Publication types

  • Comparative Study
  • English Abstract

MeSH terms

  • Administration, Cutaneous
  • Alpinia / chemistry*
  • Animals
  • Azepines / pharmacology*
  • Drugs, Chinese Herbal / pharmacology*
  • Fluorouracil / metabolism
  • Fluorouracil / pharmacokinetics*
  • Male
  • Mice
  • Mice, Nude
  • Oils, Volatile / isolation & purification
  • Oils, Volatile / pharmacology*
  • Plant Oils / pharmacology
  • Plants, Medicinal / chemistry
  • Skin Absorption / drug effects*

Substances

  • Azepines
  • Drugs, Chinese Herbal
  • Oils, Volatile
  • Plant Oils
  • Fluorouracil