Alleviation of PC4-mediated transcriptional repression by the ERCC3 helicase activity of general transcription factor TFIIH

J Biol Chem. 2003 Apr 25;278(17):14827-31. doi: 10.1074/jbc.M213172200. Epub 2003 Feb 17.

Abstract

Positive cofactor 4 (PC4), originally identified as a transcriptional coactivator, possesses the ability to suppress promoter-driven as well as nonspecific transcription via its DNA binding activity. Previous studies showed that the repressive activity of PC4 on promoter-driven transcription is alleviated by transcription factor TFIIH, possibly through one of its enzymatic activities. Using recombinant TFIIH, we have analyzed the role of TFIIH for alleviating PC4-mediated transcriptional repression and determined that the excision repair cross complementing (ERCC3) helicase activity of TFIIH is the enzymatic activity that alleviates PC4-mediated repression via beta-gamma bond hydrolysis of ATP. In addition, the alleviation does not require either ERCC2 helicase or cyclin-dependent kinase 7 kinase activity. We also show that, as complexed within TFIIH, the cyclin-dependent kinase 7 kinase does not possess the activity to phosphorylate PC4. Thus, TFIIH appears to protect promoters from PC4-mediated repression by relieving the topological constraint imposed by PC4 through the ERCC3 helicase activity rather than by reducing the repressive activity of PC4 via its phosphorylation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Cyclin-Dependent Kinase-Activating Kinase
  • Cyclin-Dependent Kinases
  • DNA Helicases / genetics*
  • DNA-Binding Proteins*
  • Humans
  • Hydrolysis
  • Immediate-Early Proteins
  • Membrane Proteins
  • Mutation
  • Phosphorylation
  • Proteins
  • Recombinant Proteins
  • Repressor Proteins / genetics*
  • Repressor Proteins / metabolism
  • Trans-Activators / genetics*
  • Trans-Activators / metabolism
  • Transcription Factor TFIIH
  • Transcription Factors*
  • Transcription Factors, TFII / genetics*
  • Transcription, Genetic*
  • Xeroderma Pigmentosum Group D Protein

Substances

  • DNA-Binding Proteins
  • IFRD2 protein, human
  • Immediate-Early Proteins
  • Membrane Proteins
  • Proteins
  • Recombinant Proteins
  • Repressor Proteins
  • Trans-Activators
  • Transcription Factors
  • Transcription Factors, TFII
  • XPBC-ERCC-3 protein
  • Transcription Factor TFIIH
  • Adenosine Triphosphate
  • Cyclin-Dependent Kinases
  • DNA Helicases
  • Xeroderma Pigmentosum Group D Protein
  • ERCC2 protein, human
  • Cyclin-Dependent Kinase-Activating Kinase
  • CDK7 protein, human