Effect of long-term oral pretreatment with levosimendan on cardiac arrhythmias during coronary artery occlusion in conscious rats

Eur J Pharmacol. 2003 Mar 19;464(2-3):171-6. doi: 10.1016/s0014-2999(03)01423-7.

Abstract

Heart failure is frequently associated with cardiac arrhythmias. The aim of the present study was to investigate the effect of levosimendan, a new cardiotonic drug for the treatment of congestive heart failure, on experimental ischaemic arrhythmias. Acute coronary artery occlusion was produced in conscious rats 7-10 days after placement of ligature around the left main coronary artery. Acute pretreatment with levosimendan (0.2 or 0.6 mg/kg orally 1 h before coronary artery occlusion) did not influence the incidence, onset and duration of arrhythmias. Long-term pretreatment with levosimendan (0.2 or 0.6 mg/kg orally twice a day for 2 weeks) increased the survival rate (50% and 81% vs. 44% in controls) and the number of animals without any arrhythmia (37% and 31% vs. 5% in controls). The present results demonstrate that chronic oral treatment with levosimendan could be beneficial in congestive heart failure and arrhythmias resulting from regional myocardial ischaemia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Animals
  • Arrhythmias, Cardiac / etiology
  • Arrhythmias, Cardiac / mortality
  • Arrhythmias, Cardiac / prevention & control*
  • Cardiotonic Agents / pharmacology*
  • Consciousness
  • Coronary Disease / complications*
  • Dose-Response Relationship, Drug
  • Electrocardiography
  • Heart / drug effects
  • Heart / physiopathology
  • Heart Rate / drug effects
  • Hydrazones / pharmacology*
  • Male
  • Myocardial Ischemia / complications
  • Pyridazines / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Simendan
  • Time Factors

Substances

  • Cardiotonic Agents
  • Hydrazones
  • Pyridazines
  • Simendan