Genetic inactivation of Par4 results in hyperactivation of NF-kappaB and impairment of JNK and p38

EMBO Rep. 2003 Mar;4(3):307-12. doi: 10.1038/sj.embor.embor769.

Abstract

The Par4 gene was first identified in prostate cells undergoing apoptosis after androgen withdrawal. PAR4 was subsequently shown to interact with, and inhibit, atypical protein kinase C isoforms, functioning as a negative regulator of the NF-kappaB pathway. This may explain its pro-apoptotic function in overexpression experiments. To determine the physiological role of PAR4, we have derived primary embryonic fibroblasts (EFs) from Par4(-/-) mice. We show here that loss of PAR4 leads to a reduction in the ability of tumour necrosis factor-alpha (TNF-alpha) to induce apoptosis by increased activation of NF-kappaB. Consistent with recent reports demonstrating the antagonistic actions of NF-kappaB and c-Jun amino-terminal kinase (JNK) signalling, we have found that Par4(-/-) cells show a reduced activation of the sustained phase of JNK and p38 stimulation by TNF-alpha and interleukin 1. Higher levels of an anti-apoptotic JNK-inhibitor protein, X-chromosome-linked inhibitor of apoptosis, in Par4(-/-) EFs might explain the inhibition of JNK activation in these cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Embryo, Mammalian
  • Fibroblasts / physiology
  • Gene Expression Regulation
  • Interleukin-1 / pharmacology
  • JNK Mitogen-Activated Protein Kinases
  • MAP Kinase Signaling System / genetics
  • Mice
  • Mice, Knockout
  • Mitogen-Activated Protein Kinases / metabolism*
  • NF-kappa B / metabolism*
  • Receptors, Thrombin / deficiency*
  • Receptors, Thrombin / genetics
  • Receptors, Thrombin / physiology*
  • Restriction Mapping
  • Tumor Necrosis Factor-alpha / pharmacology
  • X Chromosome
  • p38 Mitogen-Activated Protein Kinases

Substances

  • Interleukin-1
  • NF-kappa B
  • Receptors, Thrombin
  • Tumor Necrosis Factor-alpha
  • JNK Mitogen-Activated Protein Kinases
  • Mitogen-Activated Protein Kinases
  • p38 Mitogen-Activated Protein Kinases
  • protease-activated receptor 4