The direct interaction of phospholipase C-gamma 1 with phospholipase D2 is important for epidermal growth factor signaling

J Biol Chem. 2003 May 16;278(20):18184-90. doi: 10.1074/jbc.M208438200. Epub 2003 Mar 19.

Abstract

The epidermal growth factor (EGF) receptor has an important role in cellular proliferation, and the enzymatic activity of phospholipase C (PLC)-gamma1 is regarded to be critical for EGF-induced mitogenesis. In this study, we report for the first time a phospholipase complex composed of PLC-gamma1 and phospholipase D2 (PLD2). PLC-gamma1 is co-immunoprecipitated with PLD2 in COS-7 cells. The results of in vitro binding analysis and co-immunoprecipitation analysis in COS-7 cells show that the Src homology (SH) 3 domain of PLC-gamma1 binds to the proline-rich motif within the Phox homology (PX) domain of PLD2. The interaction between PLC-gamma1 and PLD2 is EGF stimulation-dependent and potentiates EGF-induced inositol 1,4,5-trisphosphate (IP(3)) formation and Ca(2+) increase. Mutating Pro-145 and Pro-148 within the PX domain of PLD2 to leucines disrupts the interaction between PLC-gamma1 and PLD2 and fails to potentiate EGF-induced IP(3) formation and Ca(2+) increase. However, neither PLD2 wild type nor PLD2 mutant affects the EGF-induced tyrosine phosphorylation of PLC-gamma1. These findings suggest that, upon EGF stimulation, PLC-gamma1 directly interacts with PLD2 and this interaction is important for PLC-gamma1 activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Motifs
  • Animals
  • COS Cells
  • Calcium / metabolism
  • Cell Division
  • Dose-Response Relationship, Drug
  • Epidermal Growth Factor / metabolism*
  • Glutathione / metabolism
  • Humans
  • Immunoblotting
  • Inositol 1,4,5-Trisphosphate / metabolism
  • Mutation
  • Phospholipase C gamma
  • Phospholipase D / chemistry
  • Phospholipase D / metabolism*
  • Phosphorylation
  • Precipitin Tests
  • Proline / chemistry
  • Protein Binding
  • Protein Structure, Tertiary
  • Rats
  • Recombinant Fusion Proteins / metabolism
  • Signal Transduction
  • Transfection
  • Type C Phospholipases / chemistry
  • Type C Phospholipases / metabolism*
  • Tyrosine / metabolism
  • src Homology Domains

Substances

  • Recombinant Fusion Proteins
  • Tyrosine
  • Epidermal Growth Factor
  • Inositol 1,4,5-Trisphosphate
  • Proline
  • Type C Phospholipases
  • phospholipase D2
  • Phospholipase C gamma
  • Phospholipase D
  • Glutathione
  • Calcium