Subthreshold doses of nebulized prostacyclin and rolipram synergistaically protect against lung ischemia-reperfusion

Transplantation. 2003 Mar 27;75(6):814-21. doi: 10.1097/01.TP.0000053751.22207.4E.

Abstract

Background: Pulmonary edema caused by increased microvascular permeability is an important feature of lung ischemia-reperfusion (I/R) injury.

Methods: We investigated the impact of co-aerosolized prostaglandin (PG)I(2) and the 3',5-cyclic adenosine monophosphate (cAMP)-specific phosphodiesterase inhibitor rolipram on microvascular leakage following I/R injury. Buffer-perfused rabbit lungs were exposed to 270 minutes of warm ischemia while anoxic ventilation and a positive intravascular pressure were maintained.

Results: On reperfusion, a massive increase of the capillary filtration coefficient and severe edema formation were noted, whereas microvascular pressures displayed only minor changes. Short-time aerosolization of subthreshold doses of either rolipram (33 microg) or PGI(2) (2.6 microg) at the beginning of ischemia did not attenuate the leakage response, whereas the co-aerosolization of both agents largely blocked any permeability increase and edema formation, independent of hemodynamic effects. The same was true when the co-aerosolization was undertaken before onset of ischemia. Similarly, the intravascular administration of rolipram and PGI(2) showed a synergistic reduction of I/R-induced vascular leak but demanded 10-fold higher doses. Intravascular release of cAMP was markedly enhanced on combined PGI(2)-rolipram administration but depended on the mode of delivery of these agents.

Conclusions: Low doses of aerosolized prostacyclin and rolipram synergistically protect against severe lung I/R injury and can be used independently of lung perfusion. This strategy may be suitable for an improvement of organ preservation in lung transplantation including early management of non-heart-beating donors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Capillary Permeability / drug effects
  • Cyclic AMP / metabolism
  • Disease Models, Animal
  • Drug Synergism
  • Epoprostenol / pharmacology*
  • Female
  • Lung Transplantation*
  • Male
  • Microcirculation / drug effects
  • Nebulizers and Vaporizers
  • Phosphodiesterase Inhibitors / pharmacology*
  • Platelet Aggregation Inhibitors / pharmacology*
  • Pulmonary Circulation / drug effects
  • Pulmonary Wedge Pressure / drug effects
  • Rabbits
  • Reperfusion Injury / drug therapy*
  • Reperfusion Injury / prevention & control
  • Rolipram / pharmacology*
  • Weight Gain / drug effects

Substances

  • Phosphodiesterase Inhibitors
  • Platelet Aggregation Inhibitors
  • Epoprostenol
  • Cyclic AMP
  • Rolipram