Gill (Na+,K+)-ATPase from the blue crab Callinectes danae: modulation of K+-phosphatase activity by potassium and ammonium ions

Comp Biochem Physiol B Biochem Mol Biol. 2003 Apr;134(4):631-40. doi: 10.1016/s1096-4959(03)00024-1.

Abstract

The kinetic properties of a microsomal gill (Na(+),K(+))-ATPase from the blue crab Callinectes danae were analyzed using the substrate p-nitrophenylphosphate. The (Na(+),K(+))-ATPase hydrolyzed PNPP obeying cooperative kinetics (n=1.5) at a rate of V=125.4+/-7.5 U mg(-1) with K(0.5)=1.2+/-0.1 mmol l(-1); stimulation by potassium (V=121.0+/-6.1 U mg(-1); K(0.5)=2.1+/-0.1 mmol l(-1)) and magnesium ions (V=125.3+/-6.3 U mg(-1); K(0.5)=1.0+/-0.1 mmol l(-1)) was cooperative. Ammonium ions also stimulated the enzyme through site-site interactions (n(H)=2.7) to a rate of V=126.1+/-4.8 U mg(-1) with K(0.5)=13.7+/-0.5 mmol l(-1). However, K(+)-phosphatase activity was not stimulated further by K(+) plus NH(4)(+) ions. Sodium ions (K(I)=36.7+/-1.7 mmol l(-1)), ouabain (K(I)=830.3+/-42.5 micromol l(-1)) and orthovanadate (K(I)=34.0+/-1.4 nmol l(-1)) completely inhibited K(+)-phosphatase activity. The competitive inhibition by ATP (K(I)=57.2+/-2.6 micromol l(-1)) of PNPPase activity suggests that both substrates are hydrolyzed at the same site on the enzyme. These data reveal that the K(+)-phosphatase activity corresponds strictly to a (Na(+),K(+))-ATPase in C. danae gill tissue. This is the first known kinetic characterization of K(+)-phosphatase activity in the portunid crab C. danae and should provide a useful tool for comparative studies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Binding Sites
  • Brachyura / enzymology*
  • Decapoda / enzymology
  • Gills / enzymology*
  • Kinetics
  • Microsomes / enzymology
  • Nitrophenols / metabolism
  • Organophosphorus Compounds / metabolism
  • Ouabain / pharmacology
  • Potassium / pharmacology*
  • Quaternary Ammonium Compounds / pharmacology*
  • Sodium-Potassium-Exchanging ATPase / drug effects
  • Sodium-Potassium-Exchanging ATPase / metabolism*
  • Vanadates / pharmacology

Substances

  • Nitrophenols
  • Organophosphorus Compounds
  • Quaternary Ammonium Compounds
  • nitrophenylphosphate
  • Vanadates
  • Ouabain
  • Sodium-Potassium-Exchanging ATPase
  • Potassium