Ibuprofen and acetaminophen: effect on muscle inflammation after eccentric exercise

Med Sci Sports Exerc. 2003 Jun;35(6):892-6. doi: 10.1249/01.MSS.0000069917.51742.98.

Abstract

Purpose: We examined the influence of ibuprofen and acetaminophen on muscle neutrophil and macrophage concentrations after novel eccentric contractions.

Methods: Twenty-four males (25 +/- 3 yr) were divided into three groups that received the maximal over-the-counter dose of either ibuprofen (1200 mg x d-1), acetaminophen (4000 mg x d-1), or a placebo after eccentric contractions of the knee extensors. Biopsies from the vastus lateralis were taken before and 24 h after exercise. Inflammatory cells were quantified in muscle cross-sections using immunohistochemistry.

Results: Macrophage concentrations were elevated by 1.5- to 2.5-fold (P < 0.05) at 24 h postexercise relative to preexercise concentrations, whereas neutrophil concentrations were not significantly elevated. Muscle inflammatory cell concentrations were unaffected by treatment with ibuprofen or acetaminophen when compared with placebo.

Conclusions: Maximal over-the-counter doses of ibuprofen or acetaminophen, when administered therapeutically, do not affect muscle concentrations of neutrophils or macrophages 24 h after a novel bout of eccentric contractions.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acetaminophen / administration & dosage
  • Acetaminophen / pharmacology*
  • Administration, Oral
  • Adult
  • Analgesics, Non-Narcotic / pharmacology*
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Double-Blind Method
  • Exercise*
  • Female
  • Humans
  • Ibuprofen / administration & dosage
  • Ibuprofen / pharmacology*
  • Inflammation*
  • Macrophages
  • Male
  • Muscle, Skeletal / pathology*
  • Neutrophils

Substances

  • Analgesics, Non-Narcotic
  • Anti-Inflammatory Agents, Non-Steroidal
  • Acetaminophen
  • Ibuprofen