A chimeric analog of human and salmon calcitonin eliminates antigenicity and reduces gastrointestinal disturbances

Endocrinology. 1992 Dec;131(6):2885-90. doi: 10.1210/endo.131.6.1280207.

Abstract

The minimum region in salmon calcitonin (sCT) which induces antigenicity and gastrointestinal disturbances has been identified by examining the cross-reactivity of several sCT fragments and CT analogs with antisera from sCT-treated patients, and by examining inhibition of gastrointestinal motility of these sCT fragments and CT analogs in conscious dogs. Sixteen residues at the N-terminus of sCT comprised the minimum fragment capable of inducing both activities. Human CT (hCT) showed no antigenicity and a four-order weaker inhibition of gastrointestinal motility than sCT. Based on these data, we synthesized the human and salmon chimeric CT, ACT-15, in which the 16 N-terminal residues were those of hCT and the 16 C-terminal residues were those of sCT. ACT-15 had no cross-reactivity with the antisera and had almost the same weak gastrointestinal inhibition effect as hCT in dog and rat models. Nevertheless, it retained a hypocalcemic activity and an analgesic activity comparable to sCT. These results suggest that the amino acid residues in the N-terminal half of CT are responsible for the formation of antibodies and the induction of gastrointestinal disturbances, but may not influence calcium metabolism or analgesia. Clinical studies of ACT-15 will be needed to confirm this hypothesis.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Calcitonin / adverse effects
  • Calcitonin / immunology
  • Calcitonin / pharmacology*
  • Dogs
  • Eating / drug effects
  • Epitopes / chemistry
  • Epitopes / immunology*
  • Female
  • Gastrointestinal Diseases / chemically induced
  • Gastrointestinal Diseases / prevention & control*
  • Gastrointestinal Motility / drug effects
  • Humans
  • Kinetics
  • Male
  • Molecular Sequence Data
  • Peptide Fragments / chemistry
  • Peptide Fragments / pharmacology*
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Epitopes
  • Peptide Fragments
  • salmon calcitonin
  • Calcitonin