The role of Ink4a/Arf in ErbB2 mammary gland tumorigenesis

Cancer Res. 2003 Jun 15;63(12):3395-402.

Abstract

Most human tumors display inactivation of the p53 and the p16(INK4)/pRb pathway. The Ink4a/alternative reading frame (ARF) locus encodes the p16(INK4a) and p14(ARF) (murine p19(ARF)) proteins. p16(INK4a) is deleted in 40-60% of breast cancer cell lines, and p16(INK4a) inactivation by DNA methylation occurs in < or =30% of human breast cancers. In mice genetically heterozygous for p16(INK4a) or Ink4a/Arf, predisposition to specific tumor types is enhanced. Ink4a/Arf(+/-) mice have increased E micro -Myc-induced lymphomagenesis and epidermal growth factor receptor-induced gliomagenesis. ErbB2 (epidermal growth factor receptor-related protein B2) is frequently overexpressed in human breast cancer and is sufficient for mammary tumorigenesis in vivo. We determined the role of heterozygosity at the Ink4a/Arf locus in ErbB2-induced mammary tumorigenesis. Compared with mouse mammary tumor virus-ErbB2 Ink4a/Arf(+/-) mice, mouse mammary tumor virus-ErbB2 Ink4a/Arf(wt) mammary tumors showed increased p16(INK4a), reduced Ki-67 expression, and reduced cyclin D1 protein but increased mammary tumor apoptosis with no significant change in the risk of developing mammary tumors. These studies demonstrate the contribution of Ink4a/Arf heterozygosity to tumor progression is tissue specific in vivo. In view of the important role of Ink4a/Arf in response to chemotherapy, these transgenic mice may provide a useful model for testing breast tumor therapies.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenocarcinoma / pathology
  • Aneuploidy
  • Animals
  • Apoptosis
  • Breast Neoplasms / pathology
  • Cell Cycle
  • Cell Transformation, Neoplastic / genetics*
  • Cell Transformation, Viral / genetics
  • Crosses, Genetic
  • Cyclin D1 / biosynthesis
  • Cyclin D1 / genetics
  • Cyclin-Dependent Kinase Inhibitor p16 / physiology*
  • Female
  • Gene Expression Regulation, Neoplastic
  • Genes, erbB-2*
  • Genes, p16*
  • Genetic Predisposition to Disease
  • Heterozygote
  • Humans
  • Ki-67 Antigen / biosynthesis
  • Ki-67 Antigen / genetics
  • Mammary Neoplasms, Experimental / genetics*
  • Mammary Neoplasms, Experimental / pathology
  • Mammary Tumor Virus, Mouse / physiology
  • Mice
  • Mice, Knockout
  • Mice, Transgenic
  • Organ Specificity
  • Transfection
  • Tumor Suppressor Protein p14ARF / physiology*

Substances

  • Cdkn2a protein, mouse
  • Cyclin-Dependent Kinase Inhibitor p16
  • Ki-67 Antigen
  • Tumor Suppressor Protein p14ARF
  • Cyclin D1