The serine/threonine kinase Pim-2 is a transcriptionally regulated apoptotic inhibitor

Genes Dev. 2003 Aug 1;17(15):1841-54. doi: 10.1101/gad.1105003. Epub 2003 Jul 17.

Abstract

Growth factor withdrawal results in the termination of factor-dependent transcription. One transcript that declines rapidly following growth factor deprivation of hematopoietic cells is the serine/threonine kinase pim-2. When constitutively expressed, Pim-2 conferred long-term resistance to a variety of apoptotic stimuli including growth factor withdrawal and endogenous levels of Pim-2 contributed to growth factor-mediated apoptotic resistance. Pim-2 expression maintained cell size and mitochondrial potential independently of the PI3K/Akt/TOR pathway. Pim-2-dependent maintenance of cell size and survival correlated with its ability to maintain rapamycin-resistant phosphorylation of the translational repressor 4E-BP1 and phosphorylation of the BH3 protein BAD. These results establish Pim-2 as a direct link between growth factor-induced transcription and a novel, kinase-dependent pathway that promotes cell-autonomous survival.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibiotics, Antineoplastic / pharmacology
  • Apoptosis*
  • Blotting, Northern
  • Blotting, Western
  • Cell Division
  • Cell Line
  • Cell Survival
  • Dose-Response Relationship, Drug
  • Flow Cytometry
  • Gene Expression Regulation
  • Genetic Vectors
  • Glucose / metabolism
  • Glucose / pharmacology
  • Interleukin-3 / metabolism
  • Lactates / metabolism
  • Membrane Potentials
  • Mice
  • Mitochondria / metabolism
  • Oligonucleotide Array Sequence Analysis
  • Phenotype
  • Phosphorylation
  • Plasmids / metabolism
  • Protein Serine-Threonine Kinases*
  • Proto-Oncogene Proteins / metabolism
  • Proto-Oncogene Proteins / physiology*
  • Recombinant Proteins / metabolism
  • Signal Transduction
  • Sirolimus / pharmacology
  • Staurosporine / pharmacology
  • Thapsigargin / pharmacology
  • Time Factors
  • Transcription, Genetic*
  • Transgenes

Substances

  • Antibiotics, Antineoplastic
  • Interleukin-3
  • Lactates
  • Pim2 protein, mouse
  • Proto-Oncogene Proteins
  • Recombinant Proteins
  • Thapsigargin
  • Protein Serine-Threonine Kinases
  • Staurosporine
  • Glucose
  • Sirolimus