Analysis of optically active compounds using conventional chromatography with a circular dichroism detector

J Pharm Biomed Anal. 2003 Aug 8;32(4-5):905-12. doi: 10.1016/s0731-7085(03)00192-4.

Abstract

Analysis of optically active compounds in complex samples is often based on chiral chromatography or capillary electrophoresis in order to separate the enantiomers. This requires a chiral reagent, when using conventional chromatography, or an expensive chiral column, or a chiral selector, when using capillary electrophoresis. The type of column, reagent, or additive depends highly on the compound to be analysed. A simple and generally applicable method is using a conventional HPLC column coupled to a CD detector. Separation of enantiomers is not required, as they can be identified by a positive or negative peak. A racemate does not produce a peak; neither does an optically inactive compound. The application of HPLC-CD for the identification of pharmacologically active compounds, such as dexamphetamine, 5-hydroxytryptophan, (-)-huperzine A, and interferon, as standards, in registered drugs, in falsifications, and in food supplements is described.

MeSH terms

  • Chromatography, High Pressure Liquid / methods
  • Circular Dichroism / methods*
  • Optical Rotation
  • Pharmaceutical Preparations / analysis*
  • Pharmaceutical Preparations / chemistry*

Substances

  • Pharmaceutical Preparations