The effects of caffeic acid phenethyl ester on tissue damage in lung after hindlimb ischemia-reperfusion

Pharmacol Res. 2003 Oct;48(4):397-403. doi: 10.1016/s1043-6618(03)00156-7.

Abstract

Aim: The aim of this study was to investigate the effects of caffeic acid phenethyl ester (CAPE) on the lungs as a remote organ after performing hindlimb ischemia-reperfusion (I/R) and by assessing biochemical and histopathological analysis.

Methods: The animals were divided into three groups: control, I/R, and I/R with CAPE. I/R period for 8 h was performed on the right hindlimb of all the anesthesied rats in I/R and CAPE with I/R group. In the CAPE with I/R group, the animals received CAPE 10 microM by intraperitoneal injection 1h before the reperfusion. The animals in the control and I/R groups received a similar volume of saline solution by means of intraperitoneal injection. At the end of the reperfusion period, a midsternotomy was performed. Blood, bronchoalveolar lavage (BAL) and lung tissue were obtained, and were used for biochemical and histopathological examination.

Results: The tissue and serum malondyaldehyde levels were significantly lower in the control (P=0.0001 and 0.001, respectively) and in the CAPE with I/R groups (P=0.0001 and 0.003, respectively) compared to the I/R group. Tissue Na(+)-K(+) ATPase activity in the CAPE with I/R group was significantly higher than in the I/R group (P=0.0001). Reduced activity was found in the I/R group compared to the control group (P=0.0001). Myeloperoxidase activity (P=0.001) and protein concentration (P=0.034) in BAL were significantly reduced in CAPE-treated animals when compared with the I/R group. A decreased activity and protein concentration were found in the control group compared to the I/R group (P=0.0001 and 0.024, respectively). The lungs of the I/R group displayed intense peribronchial and perivascular leukocytic infiltration in histopathological examination compared to the CAPE with I/R group (P<0.05).

Conclusion: CAPE seems to be effective in protecting remote organ injury caused by increased oxidative stress and neutrophil accumulation that results from an I/R injury.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Bronchoalveolar Lavage / methods
  • Bronchoalveolar Lavage Fluid / chemistry
  • Bronchoalveolar Lavage Fluid / cytology
  • Caffeic Acids / administration & dosage
  • Caffeic Acids / pharmacokinetics
  • Caffeic Acids / therapeutic use*
  • Capillary Permeability / drug effects
  • Hindlimb / blood supply*
  • Hindlimb / injuries*
  • Hindlimb / physiopathology
  • Injections, Intraperitoneal
  • Lung / chemistry
  • Lung / drug effects*
  • Lung / ultrastructure
  • Male
  • Malondialdehyde / antagonists & inhibitors
  • Malondialdehyde / blood
  • Neutrophil Infiltration / drug effects
  • Peroxidase / antagonists & inhibitors
  • Peroxidase / chemistry
  • Peroxidase / drug effects
  • Phenylethyl Alcohol / administration & dosage
  • Phenylethyl Alcohol / analogs & derivatives*
  • Phenylethyl Alcohol / pharmacokinetics
  • Phenylethyl Alcohol / therapeutic use*
  • Proteins / antagonists & inhibitors
  • Proteins / chemistry
  • Rats
  • Rats, Wistar
  • Reperfusion Injury / complications*
  • Reperfusion Injury / drug therapy*
  • Reperfusion Injury / physiopathology
  • Respiratory Distress Syndrome / complications*
  • Respiratory Distress Syndrome / drug therapy*
  • Respiratory Distress Syndrome / physiopathology
  • Sodium-Potassium-Exchanging ATPase / antagonists & inhibitors
  • Sodium-Potassium-Exchanging ATPase / chemistry
  • Sodium-Potassium-Exchanging ATPase / drug effects
  • Time Factors
  • Tourniquets / adverse effects
  • Turkey

Substances

  • Caffeic Acids
  • Proteins
  • Malondialdehyde
  • Peroxidase
  • Sodium-Potassium-Exchanging ATPase
  • caffeic acid phenethyl ester
  • Phenylethyl Alcohol