Cell type- and promoter-specific roles of Ser18 phosphorylation in regulating p53 responses

J Biol Chem. 2003 Oct 17;278(42):41028-33. doi: 10.1074/jbc.M306938200. Epub 2003 Aug 8.

Abstract

Phosphorylation of mouse p53 at Ser18 occurs after DNA damage. To determine the physiological roles of this phosphorylation event in p53-dependent DNA damage responses, a Ser18 to Ala missense mutation was introduced into the germline of mice. Thymocytes and fibroblasts from the knock-in mice show reduced transactivation of many p53 target genes following DNA damage. p53 protein stabilization and DNA binding are similar in knock-in and wild type mice, but C-terminal acetylation was defective, consistent with a role for Ser18 in the recruitment of transcriptional co-activators. The apoptotic response of knock-in thymocytes to ionizing radiation is intermediate between that of wild type and p53 null thymocytes. Despite impaired transcriptional and apoptotic responses, the knock-in mice are not prone to spontaneous tumorigenesis. This indicates that neither phosphorylation of p53 on Ser18 by ATM nor a full transcriptional response is essential to prevent spontaneous tumor formation in mice.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Apoptosis
  • Ataxia Telangiectasia Mutated Proteins
  • Blotting, Western
  • Cell Cycle
  • Cell Cycle Proteins
  • Chromatin / metabolism
  • DNA Damage
  • DNA-Binding Proteins
  • Dose-Response Relationship, Radiation
  • Fibroblasts / metabolism
  • Mice
  • Mice, Transgenic
  • Oligonucleotide Array Sequence Analysis
  • Phosphorylation
  • Precipitin Tests
  • Promoter Regions, Genetic*
  • Protein Serine-Threonine Kinases / metabolism
  • Protein Structure, Tertiary
  • RNA, Messenger / metabolism
  • Reverse Transcriptase Polymerase Chain Reaction
  • Serine / chemistry*
  • Serine / metabolism
  • Thymus Gland / cytology
  • Thymus Gland / metabolism
  • Time Factors
  • Transcription, Genetic
  • Transcriptional Activation
  • Tumor Suppressor Protein p53 / metabolism
  • Tumor Suppressor Proteins
  • Ultraviolet Rays

Substances

  • Cell Cycle Proteins
  • Chromatin
  • DNA-Binding Proteins
  • RNA, Messenger
  • Tumor Suppressor Protein p53
  • Tumor Suppressor Proteins
  • Serine
  • Ataxia Telangiectasia Mutated Proteins
  • Atm protein, mouse
  • Protein Serine-Threonine Kinases